SCHEMBL9328857

SCHEMBL9328857

O=C1CCCCC1c1cncc2ccccc12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.37
CYP11B2 P19099 4/20 0.37
MCL1 Q07820 1/20 0.36
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
MAPT P10636 2/20 0.35
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2B6 P20813 1/20 0.34
CYP2C19 P33261 1/20 0.34
TLR4 O00206 1/20 0.34
PLA2G6 O60733 3/20 0.34
NPC1 O15118 2/20 0.34
MAPK1 P28482 2/20 0.34
RAB9A P51151 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
FAAH O00519 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15874844 0.81 IDO1 (0.50) MCL1MAPTCYP2D6CYP2C9CYP2C19
SCHEMBL4800917 0.81 IDO1 (0.50) MCL1MAPTCYP2D6CYP2C9CYP2C19
SCHEMBL4802338 0.76 IDO1 (0.51) MAPTCYP2D6CYP2C9CYP2C19PLA2G6
SCHEMBL28442398 0.76 TDP1 (0.41) CYP11B1CYP11B2CNR1CNR2ADRA2A
SCHEMBL11665783 0.74 TDP1 (0.44) CYP11B1CYP11B2CNR1CNR2ADRA2A
Cyclohexane SCHEMBL22288135 0.74 TDP1 (0.44) CYP11B1CYP11B2CNR1CNR2ADRA2A
SCHEMBL30834543 0.72 IKBKB (0.38) CYP11B1CYP11B2CNR1CNR2MAPT
SCHEMBL21733703 0.72 IKBKB (0.38) CYP11B1CYP11B2CNR1CNR2MAPT
SCHEMBL13997857 0.72 CYP1B1 (0.42) MCL1MAPTCYP2D6CYP2C9CYP2C19
SCHEMBL21722167 0.72 GAA (0.43) MAPTMAPK1SMN1; SMN2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3746436-A1 FUSED RING COMPOUNDS F. Hoffmann-La Roche AG (CH) 2020-12-09 EP disclosed
WO-2020035031-A1 FUSED RING COMPOUNDS GENENTECH, INC. (US) 2020-02-20 WO disclosed
EP-0321274-B1 Derivatives of thioformamide MAY & BAKER LTD (GB) 1994-03-30 EP disclosed
US-5151436-A Compounds for inhibiting hair loss in men RHONE-POULENC SANTE (FR) 1992-09-29 US disclosed
EP-0321274-A1 Derivatives of thioformamide RHONE POULENC RORER LIMITED (GB) 1989-06-21 EP disclosed