SCHEMBL9329970

SCHEMBL9329970

CCn1c(=O)c(=O)[nH]c2cnccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.51
GRIA2 P42262 1/20 0.51
GRIA3 P42263 1/20 0.51
GRIA4 P48058 1/20 0.51
KDM5A P29375 5/20 0.49
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KDM5B Q9UGL1 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
KMT2A Q03164 1/20 0.41
PARP1 P09874 1/20 0.41
THRB P10828 1/20 0.40
HPGD P15428 1/20 0.40
BRPF1 P55201 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9433339 0.79 GRIA1 (0.47) GRIA1GRIA2GRIA3GRIA4KDM5A
SCHEMBL29579885 0.77 CYP1A2 (0.69) GRIA1GRIA2GRIA3GRIA4KDM4E
SCHEMBL982104 0.77 CYP1A2 (0.69) GRIA1GRIA2GRIA3GRIA4KDM4E
SCHEMBL8247664 0.75 ADORA3 (0.51) ALDH1A1MAPTSMN1; SMN2ADORA3ADORA2A
SCHEMBL4036186 0.71 PARP1 (0.42) KDM5AKDM5BPARP1GABRA5DAO
SCHEMBL2270268 0.71 CYP1A2 (0.60) KDM5ASMN1; SMN2ADORA3ADORA2AADORA1
SCHEMBL9432802 0.71 OPRL1 (0.49) PARP1METAP2DAO
SCHEMBL9106684 0.70 PARP1 (0.65) ALDH1A1PARP1DAO
SCHEMBL30363017 0.70 PARP1 (0.65) ALDH1A1PARP1DAO
SCHEMBL8609163 0.70 GRIA1 (0.65) GRIA1GRIA2GRIA3GRIA4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0589914-A1 NOVEL 3-FUSED PYRIDINIUMMETHYL CEPHALOSPORINS CHEIL FOODS & CHEMICALS, INC. (KR) 1994-04-06 EP disclosed
US-5281589-A Pharmaceuticals CHEIL FOODS & CHEMICALS, INC. (KR) 1994-01-25 US disclosed
WO-1992022556-A1 NOVEL 3-FUSED PYRIDINIUMMETHYL CEPHALOSPORINS CHEIL FOODS & CHEMICALS, INC. (KR) 1992-12-23 WO disclosed