SCHEMBL9332010

SCHEMBL9332010

C[C@@H](C(=O)O)N1c2ccccc2Sc2ccc(C#N)cc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 8/20 0.45
LMNA P02545 4/20 0.43
HTR1A P08908 2/20 0.43
DRD3 P35462 2/20 0.43
MAPK1 P28482 2/20 0.43
PGR P06401 1/20 0.43
CHRM2 P08172 1/20 0.43
ADRA2A P08913 1/20 0.43
CHRM1 P11229 1/20 0.43
DRD1 P21728 1/20 0.43
TBXA2R P21731 1/20 0.43
ACHE P22303 1/20 0.43
PTGS1 P23219 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
ADRA1A P35348 1/20 0.43
OPRM1 P35372 1/20 0.43
SLC6A3 Q01959 1/20 0.43
KCNH2 Q12809 1/20 0.43
ADRB3 P13945 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9331523 1.00 BCHE (0.45) BCHELMNAHTR1ADRD3MAPK1
SCHEMBL9759641 0.86 BCHE (0.39) BCHEACHE
SCHEMBL9759648 0.86 BCHE (0.39) BCHEACHE
SCHEMBL439056 0.84 BCHE (0.56) BCHEHTR1ADRD3ACHEPTGS1
SCHEMBL9759495 0.82 LMNA (0.43) BCHELMNAHTR1ADRD3MAPK1
SCHEMBL9331439 0.81 LMNA (0.46) BCHELMNAHTR1ADRD3MAPK1
SCHEMBL9331442 0.81 LMNA (0.46) BCHELMNAHTR1ADRD3MAPK1
SCHEMBL9331534 0.79 LMNA (0.46) BCHELMNAHTR1ADRD3MAPK1
SCHEMBL9759761 0.78 LMNA (0.43) BCHELMNAHTR1ADRD3MAPK1
SCHEMBL9759757 0.78 LMNA (0.43) BCHELMNAHTR1ADRD3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5321026-A Antispasmodic agents RHONE-POULENC RORER S.A. (FR) 1994-06-14 US disclosed
US-5049669-A Also diuretics RHONE-POULENC SANTE (FR) 1991-09-17 US disclosed
US-4985419-A Analgesics, Diuretics RHONE-POULENC SANTE (FR) 1991-01-15 US disclosed
US-4912105-A Derivatives of phenothiazine and the compositions which contain them RHONE-POULENC SANTE (FR) 1990-03-27 US disclosed