SCHEMBL933403

SCHEMBL933403

CC(C)(C)[Si](C)(C)OCCC=Cc1cccc(Br)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.38
HSD17B3 P37058 1/20 0.38
MAOA P21397 2/20 0.38
MAOB P27338 2/20 0.38
SLC6A19 Q695T7 1/20 0.37
PKM P14618 1/20 0.36
ALDH1A1 P00352 3/20 0.36
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
BACE1 P56817 1/20 0.35
IDO1 P14902 2/20 0.33
AGXT P21549 2/20 0.33
HRH4 Q9H3N8 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 2/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15539518 0.83 IDO1 (0.43) BACE1IDO1MEN1KMT2A
SCHEMBL15539516 0.83 IDO1 (0.43) BACE1IDO1MEN1KMT2A
SCHEMBL2807247 0.78 HSD17B3 (0.45) CHRNA7HSD17B3MAOAMAOBSLC6A19
SCHEMBL2807250 0.78 HSD17B3 (0.45) CHRNA7HSD17B3MAOAMAOBSLC6A19
SCHEMBL6156781 0.77 CHRNA7 (0.43) CHRNA7HSD17B3MAOAMAOBSLC6A19
SCHEMBL14833880 0.77 CHAT (0.37) ALDH1A1IDO1HRH4NPC1RAB9A
SCHEMBL14833817 0.77 CHAT (0.37) ALDH1A1IDO1HRH4NPC1RAB9A
SCHEMBL20640574 0.77 NFE2L2 (0.41) BACE1RAB9A
SCHEMBL6158612 0.74 HSP90AA1 (0.50) CHRNA7HSD17B3MAOAMAOBALDH1A1
SCHEMBL20640990 0.74 NFE2L2 (0.38) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2451793-A1 BACE INHIBITORS Eli Lilly and Company (US) 2012-05-16 EP disclosed
WO-2011005738-A1 BACE INHIBITORS ELI LILLY AND COMPANY (US) 2011-01-13 WO disclosed