SCHEMBL9336264

SCHEMBL9336264

CC(C)(C)NCC(COc1nsnc1N1CCOCC1)=NO

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.61
ADRB2 P07550 1/20 0.61
ADRB1 P08588 1/20 0.61
CYP3A4 P08684 1/20 0.61
HTR1A P08908 1/20 0.61
CYP2D6 P10635 1/20 0.61
ADRB3 P13945 1/20 0.61
NFKB1 P19838 1/20 0.61
DRD1 P21728 1/20 0.61
SIGMAR1 Q99720 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
HTT P42858 3/20 0.54
NPSR1 Q6W5P4 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.53
BLM P54132 1/20 0.53
KMT2A Q03164 5/20 0.49
MEN1 O00255 4/20 0.49
ALDH1A1 P00352 6/20 0.48
HPGD P15428 3/20 0.47
ALOX15 P16050 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9336252 1.00 CYP1A2 (0.61) CYP1A2ADRB2ADRB1CYP3A4HTR1A
Oxalic Acid SCHEMBL9336263 0.95 SMN1; SMN2 (0.56) CYP1A2ADRB2ADRB1CYP3A4HTR1A
Oxalic Acid SCHEMBL9336253 0.95 SMN1; SMN2 (0.56) CYP1A2ADRB2ADRB1CYP3A4HTR1A
SCHEMBL9337821 0.85 HTT (0.54) CYP1A2ADRB2ADRB1CYP3A4HTR1A
SCHEMBL9336258 0.85 HTT (0.54) CYP1A2ADRB2ADRB1CYP3A4HTR1A
SCHEMBL9817959 0.84 CYP1A2 (0.63) CYP1A2ADRB2ADRB1CYP3A4HTR1A
Hydrochloric Acid SCHEMBL9336231 0.84 HTT (0.53) CYP1A2ADRB2ADRB1CYP3A4HTR1A
Hydrochloric Acid SCHEMBL9336244 0.84 HTT (0.53) CYP1A2ADRB2ADRB1CYP3A4HTR1A
SCHEMBL9339905 0.82 HTT (0.60) CYP1A2ADRB2ADRB1CYP3A4HTR1A
SCHEMBL9339910 0.82 HTT (0.60) CYP1A2ADRB2ADRB1CYP3A4HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0283147-B1 Labile ketone derivatives of 3-substituted-1-alkylamino-2-propanols and their use as beta-adrenergic blockers UNIV FLORIDA (US) 1994-05-11 EP disclosed
US-5017618-A Treatment Of Glaucoma UNIVERSITY OF FLORIDA (US) 1991-05-21 US disclosed