Oxalic Acid

Oxalic Acid

SCHEMBL9342137

Cc1nc(C2=CCCNC2)co1.O=C(O)C(=O)O

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.38
SLC6A1 P30531 1/20 0.38
SLC6A13 Q9NSD5 1/20 0.38
CHRM3 P20309 4/20 0.38
CHRM2 P08172 4/20 0.38
BLM P54132 1/20 0.37
CHRM4 P08173 2/20 0.35
CHRM5 P08912 2/20 0.35
CHRM1 P11229 2/20 0.35
HTR6 P50406 1/20 0.34
ENPP3 O14638 2/20 0.33
ENPP1 P22413 1/20 0.33
PARP1 P09874 1/20 0.32
HTR2A P28223 3/20 0.32
HTR2C P28335 2/20 0.32
HTR2B P41595 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9342071 0.91 CHRM2 (0.43) CHRM3CHRM2CHRM4CHRM5CHRM1
Oxalic Acid SCHEMBL9342051 0.78 CHRM3 (0.40) TSHRSLC6A1SLC6A13CHRM3CHRM2
Oxalic Acid SCHEMBL9404337 0.75 TSHR (0.38) TSHRSLC6A1SLC6A13CHRM3CHRM2
Oxalic Acid SCHEMBL10420362 0.72 CHRM2 (0.59) TSHRSLC6A1SLC6A13CHRM3CHRM2
Oxalic Acid SCHEMBL10420357 0.72 CHRM2 (0.59) TSHRSLC6A1SLC6A13CHRM3CHRM2
Oxalic Acid SCHEMBL9342817 0.72 TSHR (0.38) TSHRSLC6A1SLC6A13CHRM3CHRM2
Oxalic Acid SCHEMBL9404449 0.69 TSHR (0.40) TSHRSLC6A1SLC6A13CHRM3CHRM2
SCHEMBL9342139 0.69 CHRM2 (0.38) CHRM3CHRM2CHRM4CHRM5CHRM1
Oxalic Acid SCHEMBL7423063 0.69 BRD4 (0.41) TSHRSLC6A1SLC6A13CHRM3CHRM2
SCHEMBL8402426 0.67 CHRM2 (0.46) CHRM3CHRM2CHRM4CHRM5CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5324723-A Analgesics MERCK SHARPE & DOHME LTD. 1994-06-28 US disclosed
EP-0307141-B1 OXAZOLES AND THIAZOLES FOR THE TREATMENT OF SENILE DEMENTIA MERCK SHARP & DOHME LTD. (GB) 1993-01-13 EP disclosed
EP-0307141-A2 Oxazoles and thiazoles for the treatment of senile dementia MERCK SHARP & DOHME LTD. (GB) 1989-03-15 EP disclosed