Glyfoline

Glyfoline

SCHEMBL9348448

COc1c(OC)c(OC)c2c(c1O)c(=O)c1ccc(O)c(OC)c1n2C

nearest known ligand 0.74

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSV O60911 8/20 0.74
MAOA P21397 5/20 0.46
KDM1A O60341 1/20 0.42
CYP19A1 P11511 2/20 0.39
PTGS2 P35354 1/20 0.39
NQO2 P16083 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Glyfoline SCHEMBL31285722 1.00 CTSV (0.74) CTSVMAOAKDM1ACYP19A1PTGS2
Citibrasine SCHEMBL9352197 0.85 CTSV (1.00) CTSVMAOAKDM1ACYP19A1KDM4E
SCHEMBL9348539 0.85 CTSV (0.68) CTSVMAOAKDM1ACYP19A1NQO2
SCHEMBL31384423 0.84 CTSV (0.76) CTSVMAOAKDM1ACYP19A1PTGS2
SCHEMBL29877319 0.81 CTSV (0.53) CTSVMAOAKDM1ACYP19A1PTGS2
SCHEMBL9348595 0.78 CTSV (0.60) CTSVMAOAKDM1ACYP19A1KDM4E
SCHEMBL9349831 0.78 CTSV (0.58) CTSVKDM1ACYP19A1NQO2ALDH1A1
SCHEMBL9348590 0.77 CTSV (0.57) CTSVKDM1ACYP19A1NQO2ALDH1A1
SCHEMBL9352227 0.76 CTSV (0.60) CTSVMAOAKDM1ACYP19A1KDM4E
Citpressine Ii SCHEMBL29711402 0.75 CTSV (0.52) CTSVMAOAKDM1AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992016509-A1 MULTISUBSTITUTED 1-HYDROXY-9-ACRIDONES WITH ANTICANCER ACTIVITY SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-10-01 WO claimed
US-5296602-A Condensing substituted ortho-halo- or ortho-aminobenzoic acid with meta-halo- or meta-aminoanisole, cyclizing, N-alkylating, de-O-methylating SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-03-22 US disclosed
WO-1992016509-A1 MULTISUBSTITUTED 1-HYDROXY-9-ACRIDONES WITH ANTICANCER ACTIVITY SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-10-01 WO disclosed