SCHEMBL9350602

SCHEMBL9350602

CCCc1cc2[nH]c(=O)ccc2c(C)n1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 3/20 0.49
PDE3A Q14432 3/20 0.49
BACE1 P56817 1/20 0.46
CYP1A2 P05177 1/20 0.43
MAPT P10636 5/20 0.42
ALDH1A1 P00352 4/20 0.41
HSD17B10 Q99714 1/20 0.41
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
GAA P10253 2/20 0.40
HPGD P15428 2/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3189390 0.77 PDE3B (0.56) PDE3BPDE3ACYP1A2MAPTALDH1A1
SCHEMBL3179823 0.72 PDE3B (0.58) PDE3BPDE3AALDH1A1SMN1; SMN2GAA
SCHEMBL8852559 0.69 DYRK1A (0.53) MAPTALDH1A1HSD17B10SMN1; SMN2GAA
SCHEMBL4306387 0.68 BACE1 (0.66) BACE1CYP1A2MAPTALDH1A1HSD17B10
SCHEMBL18932511 0.66 CA12 (0.46) PDE3BPDE3ABACE1CA12CA9
SCHEMBL10813255 0.66 PDE3B (1.00) PDE3BPDE3A
Medorinone SCHEMBL121782 0.65 PDE3B (1.00) PDE3BPDE3ACYP1A2MAPTALDH1A1
SCHEMBL27688255 0.65 PDE3B (0.54) PDE3BPDE3AALDH1A1SMN1; SMN2GAA
SCHEMBL10727584 0.65 PDE3B (0.53) PDE3BPDE3ACYP1A2MAPTALDH1A1
SCHEMBL188316 0.65 MAPK1 (0.43) PDE3BPDE3ACYP1A2ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5294620-A Hypotensive agents or compounds for cardiovascular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-03-15 US disclosed
US-5217976-A Hypotensive agents, congestive heart failure IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-06-08 US disclosed