SCHEMBL9354561

SCHEMBL9354561

Cc1ccc(S(=O)(=O)n2cnc(C[C@H](NC(=O)OC(C)(C)C)C(=O)N3CCCN3C(=O)O[C@@H](Cc3ccccc3)C(=O)O)c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KLK7 P49862 1/20 0.56
TLR2 O60603 1/20 0.46
TLR1 Q15399 1/20 0.46
P2RX7 Q99572 7/20 0.43
KMT2A Q03164 2/20 0.39
MAPK1 P28482 1/20 0.38
ALDH1A1 P00352 2/20 0.38
TSHR P16473 1/20 0.38
ACE P12821 1/20 0.37
MCL1 Q07820 2/20 0.37
HRH2 P25021 1/20 0.37
HRH1 P35367 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9354935 0.93 KLK7 (0.57) KLK7TLR2TLR1P2RX7
SCHEMBL9354881 0.90 KLK7 (0.60) KLK7TLR2TLR1P2RX7
SCHEMBL29401167 0.81 KLK7 (0.61) KLK7TLR2TLR1KMT2AALDH1A1
SCHEMBL3912355 0.81 KLK7 (0.61) KLK7TLR2TLR1KMT2AALDH1A1
SCHEMBL9354399 0.79 MAPK1 (0.58) KMT2AMAPK1ACEHRH2HRH1
SCHEMBL9354395 0.79 MAPK1 (0.58) KMT2AMAPK1ACEHRH2HRH1
SCHEMBL6163528 0.79 KLK7 (0.56) KLK7TLR2TLR1P2RX7KMT2A
SCHEMBL7441367 0.74 KLK7 (0.53) KLK7TLR2TLR1KMT2AALDH1A1
SCHEMBL3911500 0.74 KLK7 (0.57) KLK7TLR2TLR1P2RX7ALDH1A1
SCHEMBL29398857 0.73 KLK7 (0.53) KLK7TLR2TLR1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0300189-B1 New amino acid derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1994-11-02 EP disclosed
EP-0300189-A2 New amino acid derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-01-25 EP disclosed