SCHEMBL9357331

SCHEMBL9357331

c1ccc(-c2ccc(CCC3CN4CCC3CC4)cc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
EGFR P00533 1/20 0.43
POLB P06746 1/20 0.43
CHRM2 P08172 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
MAPT P10636 1/20 0.43
CHRM1 P11229 1/20 0.43
DRD2 P14416 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
CHRM3 P20309 1/20 0.43
DRD1 P21728 1/20 0.43
SLC6A2 P23975 1/20 0.43
HTR2A P28223 1/20 0.43
SLC6A4 P31645 1/20 0.43
ADRA1A P35348 1/20 0.43
HRH1 P35367 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8931451 0.98 CHRNB4 (0.42) CHRNB4CHRNA3EGFRPOLBCHRM2
SCHEMBL3215425 0.91 CHRNB4 (0.47) CHRNB4CHRNA3EGFRPOLBCHRM2
SCHEMBL8863847 0.84 CHRNB4 (0.45) CHRNB4CHRNA3EGFRPOLBCHRM2
Hydrochloric Acid SCHEMBL8864188 0.83 CHRNB4 (0.44) CHRNB4CHRNA3EGFRPOLBCHRM2
Hydrochloric Acid SCHEMBL10914610 0.80 GAA (0.55) HTR3ACYP2D6CHRNA7
SCHEMBL7330957 0.76 LTA4H (0.50) CHRM1CHRM3KCNH2
Hydrochloric Acid SCHEMBL7430573 0.75 LTA4H (0.49) CHRM1CHRM3KCNH2
SCHEMBL3214765 0.74 CHRNB4 (0.50) CHRNB4CHRNA3EGFRPOLBCHRM2
SCHEMBL13444728 0.74 CHRNB4 (0.50) CHRNB4CHRNA3EGFRPOLBCHRM2
SCHEMBL9541328 0.72 USP30 (0.52) CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626960-A1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS ZENECA LIMITED (GB) 1994-12-07 EP claimed
WO-1993013096-A1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-07-08 WO claimed
WO-1993013096-A1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-07-08 WO disclosed