SCHEMBL9358949

SCHEMBL9358949

CNCC=C(Oc1ccc(O)cc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.41
CYP19A1 P11511 5/20 0.41
ELANE P08246 7/20 0.39
DRD4 P21917 2/20 0.39
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
LTA4H P09960 1/20 0.38
NR1H2 P55055 1/20 0.38
BAX Q07812 1/20 0.38
ESRRG P62508 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
PTGS1 P23219 1/20 0.38
SLC6A2 P23975 1/20 0.38
CYP2C19 P33261 1/20 0.38
PTGS2 P35354 1/20 0.38
SLC6A3 Q01959 1/20 0.38
HIF1A Q16665 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
ESR2 Q92731 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9595848 0.94 DRD4 (0.39) ESR1CYP19A1ELANEDRD4DRD2
SCHEMBL9359225 0.91 HTR1B (0.38) ELANECYP1A2MEN1MAPTTHRB
SCHEMBL9359229 0.91 HTR1B (0.38) ELANECYP1A2MEN1MAPTTHRB
SCHEMBL9359262 0.91 HTR1B (0.38) ELANECYP1A2MEN1MAPTTHRB
SCHEMBL9363320 0.88 NPC1 (0.45) LTA4HLMNACYP1A2CYP2C19PTGS2
SCHEMBL9359049 0.87 SLC6A4 (0.40) ELANEDRD4DRD2DRD3LMNA
SCHEMBL9359074 0.84 KMT2A (0.49) ELANELMNACYP1A2NPC1MAPT
SCHEMBL9358624 0.84 CYP3A4 (0.43) ESR1DRD4DRD2DRD3ESR2
SCHEMBL9358617 0.84 CYP3A4 (0.43) ESR1DRD4DRD2DRD3ESR2
SCHEMBL9358620 0.84 CYP3A4 (0.43) ESR1DRD4DRD2DRD3ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0363782-B1 Aryloxy-, arylthio-, heteroaryloxy-, heteroarylthio-alkenylene derivatives of amines ERBA CARLO SPA (IT) 1994-01-05 EP disclosed
US-5272144-A Aryloxy-, arylthio-, heteroaryloxy-, heteroarylthio-alkenylene derivatives of amines and pharmaceutical use FARMITALIA CARLO ERBA S.R.L. (IT) 1993-12-21 US disclosed
WO-1990003965-A1 ARYLOXY-, ARYLTHIO-, HETEROARYLOXY-, HETEROARYLTHIO-ALKENYLENE DERIVATIVES OF AMINES FARMITALIA CARLO ERBA S.R.L. (IT) 1990-04-19 WO disclosed