Ethyne

Ethyne

SCHEMBL9362017

C#C.C=C1CCN(C)CC1

nearest known ligand 0.37

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.37
MAOB P27338 3/20 0.37
DRD2 P14416 3/20 0.37
DRD1 P21728 3/20 0.37
DRD5 P21918 3/20 0.37
DRD3 P35462 3/20 0.37
DRD4 P21917 1/20 0.37
NOS1 P29475 1/20 0.36
SETD7 Q8WTS6 3/20 0.33
ADRA2A P08913 1/20 0.31
CYP2D6 P10635 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31
SLC6A4 P31645 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL272823 0.94
Hydrochloric Acid SCHEMBL9869384 0.91
SCHEMBL9965402 0.83
SCHEMBL10284651 0.77
SCHEMBL22885439 0.77 INMT (0.36) MAOAMAOBDRD2DRD1DRD5
Maleic Acid SCHEMBL9877527 0.74 CYP3A4 (0.45) DRD2DRD1DRD5DRD3ADRA2A
Fumaric Acid SCHEMBL9877532 0.74 CYP3A4 (0.45) DRD2DRD1DRD5DRD3ADRA2A
SCHEMBL14409996 0.74 KDM1A (0.38) CYP2D6
SCHEMBL24811636 0.72 CHKA (0.31) MAOAMAOBDRD2DRD1DRD5
SCHEMBL22885428 0.70 INMT (0.32) DRD2DRD1DRD5DRD3DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0418143-B1 Dicarboxylic acids derivatives containing a nitrogen or oxygen heteroring, process for their preparation and their use as medicines ROUSSEL UCLAF (FR) 1994-03-23 EP claimed