SCHEMBL9364683

SCHEMBL9364683

N#Cc1cc2c(cc1C(F)(F)F)[nH]c(=O)c(=O)n2OC1CCCCC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
AR P10275 13/20 0.35
OPRM1 P35372 1/20 0.34
OPRL1 P41146 1/20 0.34
PDE9A O76083 2/20 0.33
CTSC P53634 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9365324 0.82 KDM4E (0.38) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9368415 0.78 GRIA1 (0.39) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9364703 0.76 KDM4E (0.35) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9364648 0.76 GRIA1 (0.43) KDM4E
SCHEMBL9365049 0.75 GRIA1 (0.39) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9091900 0.75 GRIA1 (0.40) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9080817 0.74 SMN1; SMN2 (0.45) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9365208 0.74 GRIA2 (0.39) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9364647 0.74 GRIA1 (0.41) ALDH1A1AR
SCHEMBL9364643 0.72 GRIA1 (0.38) KDM4EALDH1A1GLAGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0377112-B1 Quinoxaline compounds and their preparation and use NOVO NORDISK AS (DK) 1994-08-24 EP disclosed
US-5061706-A 2,3-QUINOXALINEDIONES FOR USE AS NEUROLEPTICS NOVO NORDISK A/S (DK) 1991-10-29 US disclosed
EP-0377112-A1 Quinoxaline compounds and their preparation and use NOVO NORDISK A/S (DK) 1990-07-11 EP disclosed