SCHEMBL9367277

SCHEMBL9367277

COc1ccc2cc(C(C)CN3CC=C(c4cccc(C(F)(F)F)c4)CC3)ccc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.46
PPARA Q07869 2/20 0.46
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
PLAU P00749 2/20 0.43
PLAT P00750 2/20 0.43
HTR7 P34969 3/20 0.41
ABCB11 O95342 1/20 0.39
PLG P00747 1/20 0.39
POLB P06746 1/20 0.39
PARP1 P09874 1/20 0.38
HTR1A P08908 2/20 0.38
MAOA P21397 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR6 P50406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8742185 0.99 PPARG (0.46) PPARGPPARAKDM4EALDH1A1GAA
SCHEMBL9618625 0.91 PPARG (0.45) PPARGPPARAKDM4EALDH1A1GAA
Hydrochloric Acid SCHEMBL9423232 0.90 PPARG (0.44) PPARGPPARAKDM4EALDH1A1GAA
SCHEMBL6168598 0.82 PPARG (0.42) PPARGPPARAKDM4EMAPTMEN1
SCHEMBL9366795 0.82 PPARG (0.45) PPARGPPARAKDM4EALDH1A1GAA
SCHEMBL9366389 0.81 PPARG (0.53) PPARGPPARAKDM4EALDH1A1GAA
SCHEMBL4588655 0.81 PPARG (0.51) PPARGPPARAKDM4EMAPTMEN1
SCHEMBL4589097 0.81 PPARG (0.51) PPARGPPARAKDM4EMAPTMEN1
SCHEMBL4589201 0.81 PPARG (0.51) PPARGPPARAKDM4EMAPTMEN1
Hydrochloric Acid SCHEMBL8742253 0.80 PPARG (0.53) PPARGPPARAKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458697-B1 N-substituted trifluoromethylphenyl tetrahydropyridines, process for their preparation, intermediates and pharmaceutical preparations containing them SANOFI ELF (FR) 1994-07-27 EP disclosed
EP-0458697-A1 N-substituted trifluoromethylphenyl tetrahydropyridines, process for their preparation, intermediates and pharmaceutical preparations containing them ELF SANOFI (FR) 1991-11-27 EP disclosed