SCHEMBL9369333

SCHEMBL9369333

S=c1[nH]ccn1Cc1cccs1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DBH P09172 11/20 0.56
ALDH1A1 P00352 2/20 0.56
CYP1A2 P05177 1/20 0.49
POLB P06746 1/20 0.49
CYP3A4 P08684 1/20 0.49
HPGD P15428 1/20 0.49
TSHR P16473 1/20 0.49
NFKB1 P19838 1/20 0.49
BLM P54132 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9442376 0.84 POLB (0.58) DBHALDH1A1POLB
SCHEMBL9442377 0.81 POLB (0.51) DBHALDH1A1POLB
SCHEMBL9442375 0.72 DBH (0.57) DBHALDH1A1CYP1A2POLBCYP3A4
SCHEMBL9442398 0.72 DBH (0.50) DBHALDH1A1CYP1A2POLBCYP3A4
SCHEMBL11079680 0.72 DBH (1.00) DBHALDH1A1CYP1A2POLBCYP3A4
SCHEMBL9442384 0.71 DBH (0.42) DBHALDH1A1CYP1A2POLBCYP3A4
SCHEMBL9442394 0.71 DBH (0.42) DBHALDH1A1CYP1A2POLBCYP3A4
SCHEMBL9371273 0.70 DBH (0.60) DBHALDH1A1CYP1A2POLBCYP3A4
SCHEMBL9368556 0.70 DBH (0.56) DBHALDH1A1CYP1A2POLBCYP3A4
SCHEMBL10556159 0.69 DBH (0.46) DBHALDH1A1CYP1A2POLBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0244803-B1 Novel dopamine beta hydroxylase inhibitors MERRELL DOW PHARMA (US) 1994-10-26 EP disclosed
US-5198457-A Treatment of hyperthyroidism with 1,3-dihydro-1[2-(2-thienyl)alkyl]-2H-imidazole-2-thiones MERRELL DOW PHARMACEUTICALS INC. (US) 1993-03-30 US disclosed
US-5189052-A Hypotensive agent MERRELL DOW PHARMACEUTICALS INC. (US) 1993-02-23 US disclosed
US-5057613-A Hypotensive agents MERRELL DOW PHARMACEUTICALS (US) 1991-10-15 US disclosed
US-4810800-A HYPOTENSIVE AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1989-03-07 US disclosed
EP-0244803-A2 Novel dopamine beta hydroxylase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1987-11-11 EP disclosed