SCHEMBL9375647

SCHEMBL9375647

CS(=O)(=O)OCC1COc2ccc(Cl)cc2O1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.58
CA1 P00915 1/20 0.52
FFAR1 O14842 16/20 0.50
CYP2C9 P11712 1/20 0.48
CYP2B6 P20813 1/20 0.48
SLCO1B3 Q9NPD5 1/20 0.48
HTR1A P08908 1/20 0.42
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
ADRA1D P25100 1/20 0.42
HTR2C P28335 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
DRD3 P35462 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL567448 0.84 CA2 (0.52) CA2FFAR1DRD2
SCHEMBL1044755 0.84 CA2 (0.53) CA2CA1FFAR1CYP2C9CYP2B6
SCHEMBL6980879 0.84 CA2 (0.53) CA2CA1FFAR1CYP2C9CYP2B6
SCHEMBL6740016 0.82 FFAR1 (0.51) CA2FFAR1CYP2C9CYP2B6SLCO1B3
SCHEMBL7982000 0.82 CA2 (0.55) CA2
SCHEMBL2544576 0.82 CA2 (0.55) CA2
SCHEMBL1545420 0.82 CA2 (0.55) CA2
SCHEMBL17272699 0.82 CA2 (0.53) CA2CA1FFAR1CYP2C9CYP2B6
SCHEMBL17272700 0.82 CA2 (0.53) CA2CA1FFAR1CYP2C9CYP2B6
SCHEMBL12056274 0.82 CA2 (0.65) CA2CA1FFAR1CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445026-B1 Aminomethylpiperidine derivatives, their process for preparation and the pharmaceutical compositions containing them ADIR (FR) 1994-01-26 EP disclosed
US-5229399-A Analgesics ADIR ET COMPAGNIE (FR) 1993-07-20 US disclosed
US-5229398-A Analgesics ADIR ET COMPAGNIE (FR) 1993-07-20 US disclosed
US-5192775-A Analgesics ADIR ET COMPAGNIE (FR) 1993-03-09 US disclosed
EP-0445026-A1 Aminomethylpiperidine derivatives, their process for preparation and the pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1991-09-04 EP disclosed