SCHEMBL9375722

SCHEMBL9375722

Cc1cc2cc(N(C(N)=O)c3cccc4cnccc34)ccc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.43
CYP2A6 P11509 1/20 0.36
KEAP1 Q14145 1/20 0.36
VCP P55072 3/20 0.36
TRPV1 Q8NER1 1/20 0.35
FGFR1 P11362 1/20 0.35
SRC P12931 1/20 0.35
FGFR2 P21802 1/20 0.35
FGFR4 P22455 1/20 0.35
FGFR3 P22607 1/20 0.35
CLK1 P49759 2/20 0.34
CDK5 Q00535 2/20 0.34
DYRK1A Q13627 2/20 0.34
CDK5R1 Q15078 2/20 0.34
CLK2 P49760 1/20 0.34
CLK3 P49761 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
KDM4E B2RXH2 2/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9371950 0.87 KDR (0.38) KDRCYP2A6KEAP1VCPFGFR1
SCHEMBL9371975 0.82 CYP3A4 (0.41) CYP2A6KEAP1VCPKDM4ECYP3A4
SCHEMBL9370838 0.81 VCP (0.42) CYP2A6KEAP1VCPDYRK1ADYRK1B
Hydrochloric Acid SCHEMBL7112841 0.79 VCP (0.41) CYP2A6KEAP1VCPKDM4ELMNA
SCHEMBL9544511 0.77 MAPT (0.42) TRPV1KDM4ELMNACYP1A2CYP3A4
SCHEMBL9370928 0.74 VCP (0.39) KDRCYP2A6KEAP1VCPFGFR1
SCHEMBL2359679 0.70 KDM4E (0.47) TRPV1KDM4ELMNACYP1A2CYP3A4
SCHEMBL9370533 0.69 CYP2A6 (0.38) CYP2A6KEAP1VCPKDM4EMAOA
SCHEMBL9370953 0.69 CYP2A6 (0.38) CYP2A6KEAP1VCPKDM4EMAOA
SCHEMBL28304454 0.67 KDM4E (0.46) TRPV1KDM4ELMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630373-A1 INDOLE DERIVATIVES AS 5HT1C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-12-28 EP disclosed