SCHEMBL9375877

SCHEMBL9375877

Cc1ccc(CCc2ccc(N)cc2)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GFER P55789 2/20 0.50
DHFR P00374 1/20 0.44
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2A6 P11509 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
NOS3 P29474 1/20 0.44
NOS2 P35228 1/20 0.44
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
ACHE P22303 1/20 0.41
PDE10A Q9Y233 1/20 0.40
CYP19A1 P11511 3/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
KCNH2 Q12809 1/20 0.40
AOC3 Q16853 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8269251 0.89 DHFR (0.45) DHFRCYP1A2CYP2A6TAAR1NOS3
SCHEMBL22460731 0.85 DHFR (0.43) DHFRCYP1A2CYP2A6TAAR1NOS3
SCHEMBL18682734 0.82 CCR1 (0.52) CYP2A6NOS3NOS2MEN1RAB9A
SCHEMBL20909966 0.79 MCHR1 (0.53) DHFRMAOBTAAR1RAB9AACHE
SCHEMBL657443 0.79 HRH1 (0.47) CYP1A2CYP2A6TAAR1NOS3NOS2
SCHEMBL19200847 0.79 PDE10A (0.43) DHFRCYP1A2NOS3NOS2NPC1
SCHEMBL18648928 0.79 TSHR (0.43) CYP1A2NOS3NOS2MEN1KMT2A
SCHEMBL10504713 0.78 SMN1; SMN2 (0.52) NOS3NOS2MEN1NPC1RAB9A
SCHEMBL29160674 0.78 TAAR1 (0.44) MAOBTAAR1ACHEPDE10AHTR2A
SCHEMBL19255610 0.78 GFER (0.74) GFERMAOAMAOBCYP1A2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0356234-B1 New Benzazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1994-05-11 EP disclosed
US-5047411-A Antiulcer Agents, H2-Receptor Antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-09-10 US disclosed
EP-0356234-A2 New Benzazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-02-28 EP disclosed