SCHEMBL9376353

SCHEMBL9376353

c1ccc(CSc2cnc3ccccc3n2)nc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.57
RAB9A P51151 9/20 0.57
SMN1; SMN2 Q16637 8/20 0.57
KDM4E B2RXH2 4/20 0.53
GAA P10253 2/20 0.53
CYP1A2 P05177 1/20 0.52
CYP2E1 P05181 1/20 0.52
CYP2C8 P10632 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2B6 P20813 1/20 0.52
CYP2C19 P33261 1/20 0.52
MAPT P10636 6/20 0.50
HPGD P15428 2/20 0.47
HTT P42858 2/20 0.47
ALDH1A1 P00352 2/20 0.47
POLB P06746 2/20 0.47
MAPK1 P28482 1/20 0.47
KLK7 P49862 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9695063 0.98 NPC1 (0.56) NPC1RAB9ASMN1; SMN2KDM4EGAA
Hydrochloric Acid SCHEMBL10562883 0.79 SMN1; SMN2 (0.52) NPC1RAB9ASMN1; SMN2KDM4EGAA
SCHEMBL23691408 0.77 NPC1 (0.60) NPC1RAB9ASMN1; SMN2KDM4ECYP1A2
SCHEMBL9381251 0.77 SMN1; SMN2 (0.50) NPC1RAB9ASMN1; SMN2KDM4ECYP1A2
Hydrochloric Acid SCHEMBL10564648 0.75 NPC1 (0.58) NPC1RAB9ASMN1; SMN2KDM4ECYP1A2
SCHEMBL9377015 0.75 KDM4E (0.50) NPC1RAB9ASMN1; SMN2KDM4EGAA
SCHEMBL9695261 0.73 MAPT (0.56) NPC1RAB9ASMN1; SMN2KDM4EGAA
SCHEMBL28002004 0.73 PDE10A (0.78) CYP1A2CYP2D6MAPTLMNAKMT2A
SCHEMBL19204573 0.72 NPC1 (0.51) NPC1RAB9ASMN1; SMN2KDM4EGAA
Hydrochloric Acid SCHEMBL9695852 0.72 MAPT (0.54) NPC1RAB9ASMN1; SMN2KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-1261387-A None JP disclosed
EP-0338346-B1 Quinoxaline derivatives and antiulcer agents NISSHIN FLOUR MILLING CO (JP) 1994-11-30 EP disclosed
US-5106976-A Antisecretory agents NIPPON CHEMIPHAR CO., LTD. (JP) 1992-04-21 US disclosed
EP-0234690-B1 SULFOXIDE DERIVATIVES AND THEIR PREPARATION NIPPON CHEMIPHAR CO., LTD. (JP) 1991-05-15 EP disclosed
US-4933458-A ANTISECRETORY AGENTS NIPPON CHEMIPHAR CO., LTD. (JP) 1990-06-12 US disclosed
US-4933342-A Quinoxaline derivatives and antiulcer agents NISSHIN FLOUR MILLING CO., LTD. (JP) 1990-06-12 US disclosed
EP-0338346-A2 Quinoxaline derivatives and antiulcer agents NISSHIN FLOUR MILLING CO., LTD. (JP) 1989-10-25 EP disclosed
JP-H01261387-A NOVEL QUINOXALINE DERIVATIVE AND ANTIULCER AGENT CONTAINING SAID DERIVATIVE NISSHIN FLOUR MILLING CO LTD 1989-10-18 JP disclosed
EP-0234690-A1 Sulfoxide derivatives and their preparation NIPPON CHEMIPHAR CO., LTD. (JP) 1987-09-02 EP disclosed