SCHEMBL9377286

SCHEMBL9377286

COC(=O)NC(=O)C1CCC(=O)N1C(=O)OCc1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.43
HTR2C P28335 1/20 0.42
CPB1 P15086 1/20 0.42
ALDH1A1 P00352 1/20 0.41
CYP2C19 P33261 1/20 0.41
FKBP1A P62942 1/20 0.41
PREP P48147 1/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29816738 0.86 KMT2A (0.49) SMN1; SMN2NPC1RAB9AHTTNPSR1
SCHEMBL19313922 0.86 KMT2A (0.49) SMN1; SMN2NPC1RAB9AHTTNPSR1
SCHEMBL20886535 0.86 KMT2A (0.49) SMN1; SMN2NPC1RAB9AHTTNPSR1
SCHEMBL15743850 0.86 SMN1; SMN2 (0.48) SMN1; SMN2NPC1RAB9AHTR2CALDH1A1
SCHEMBL8290690 0.86 SMN1; SMN2 (0.48) SMN1; SMN2NPC1RAB9AHTR2CALDH1A1
SCHEMBL4387495 0.84 KDM4E (0.51) SMN1; SMN2NPC1RAB9AHTTNPSR1
SCHEMBL3845188 0.83 SMN1; SMN2 (0.53) SMN1; SMN2NPC1RAB9ANPSR1HTR2C
SCHEMBL3600148 0.83 SMN1; SMN2 (0.53) SMN1; SMN2NPC1RAB9ANPSR1HTR2C
SCHEMBL3600152 0.83 SMN1; SMN2 (0.53) SMN1; SMN2NPC1RAB9ANPSR1HTR2C
SCHEMBL4388871 0.82 NPSR1 (0.56) SMN1; SMN2RAB9AHTTNPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0353778-B1 Pyrrolo[1,4]benzodiazepine derivatives SHIONOGI & CO (JP) 1994-11-02 EP disclosed
US-4923984-A TREATMENT OF SENILE DEMENTIA, PSYCHONEUROSIS, AMNESIA SHIONOGI & CO., LTD. (JP) 1990-05-08 US disclosed
EP-0353778-A2 Pyrrolo[1,4]benzodiazepine derivatives SHIONOGI & CO., LTD. (JP) 1990-02-07 EP disclosed