SCHEMBL9380384

SCHEMBL9380384

OCc1nccn1-c1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.52
PDE4A P27815 1/20 0.48
PDE4B Q07343 1/20 0.48
PDE4C Q08493 1/20 0.48
PDE4D Q08499 1/20 0.48
CYP19A1 P11511 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
MAPKAPK2 P49137 1/20 0.40
NOTUM Q6P988 4/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
BIRC5 O15392 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8364531 0.82 MAPKAPK2 (0.40) KCNH2CYP19A1MEN1ALDH1A1CYP1A2
SCHEMBL3748867 0.82 PDE4A (0.48) KCNH2PDE4APDE4BPDE4CPDE4D
SCHEMBL22310226 0.82 PDE4A (0.48) KCNH2PDE4APDE4BPDE4CPDE4D
SCHEMBL27450288 0.82 PDE4A (0.54) KCNH2PDE4APDE4BPDE4CPDE4D
SCHEMBL4314558 0.81 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL30638906 0.81 KCNH2 (0.46) KCNH2PDE4APDE4BPDE4CPDE4D
SCHEMBL243235 0.79 PDE4A (0.45) KCNH2PDE4APDE4BPDE4CPDE4D
SCHEMBL22309076 0.78 ALDH1A1 (0.49) PDE4APDE4BPDE4CPDE4DCYP19A1
SCHEMBL3746738 0.76 PDE4A (0.46) KCNH2PDE4APDE4BPDE4CPDE4D
SCHEMBL6609392 0.76 MAPKAPK2 (0.43) KCNH2CYP19A1MEN1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0289380-B1 Aryl-heteroaryl-carbinol derivatives having an analgesic activity ESTEVE LABOR DR (ES) 1994-12-28 EP claimed
WO-2016124139-A1 HETEROCYCLIC-SUBSTITUTED N-SULFONYLBENZAMIDE DERIVATIVES, PREPARATION METHOD FOR DERIVATIVES, AND PHARMACEUTICAL USE OF DERIVATIVES 上海海雁医药科技有限公司 2016-08-11 WO disclosed