SCHEMBL9384200

SCHEMBL9384200

Cc1ccc(C(=O)c2ccc3n2CCC3C(=O)O)cc1.[CaH2]

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.75
CDC42 P60953 3/20 0.75
RAC1 P63000 3/20 0.75
PTGS1 P23219 3/20 0.75
PAK1 Q13153 2/20 0.75
NPC1 O15118 1/20 0.75
CHRM3 P20309 1/20 0.75
OPRM1 P35372 1/20 0.75
RAB9A P51151 1/20 0.75
LMNA P02545 2/20 0.65
ABCC4 O15439 1/20 0.65
HTT P42858 1/20 0.65
BLM P54132 1/20 0.65
CYP1A2 P05177 1/20 0.65
NFKB1 P19838 1/20 0.65
MAPK1 P28482 1/20 0.65
CA4 P22748 5/20 0.47
CA9 Q16790 4/20 0.47
CA12 O43570 3/20 0.47
CA1 P00915 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9382190 0.99 PTGS2 (0.77) PTGS2CDC42RAC1PTGS1PAK1
SCHEMBL11601847 0.97 PTGS2 (0.75) PTGS2CDC42RAC1PTGS1PAK1
SCHEMBL11602055 0.97 PTGS2 (0.75) PTGS2CDC42RAC1PTGS1PAK1
SCHEMBL11201558 0.92 PTGS2 (0.64) PTGS2CDC42RAC1PTGS1PAK1
SCHEMBL11194044 0.91 PTGS2 (0.65) PTGS2CDC42RAC1PTGS1PAK1
SCHEMBL11206957 0.90 PTGS2 (0.64) PTGS2CDC42RAC1PTGS1PAK1
SCHEMBL11197740 0.90 PTGS2 (0.64) PTGS2CDC42RAC1PTGS1PAK1
SCHEMBL11198770 0.90 PTGS2 (0.64) PTGS2CDC42RAC1PTGS1PAK1
Ketorolac SCHEMBL28092302 0.87 PTGS2 (0.97) PTGS2CDC42RAC1PTGS1PAK1
P-Hydroxy Ketorolac SCHEMBL17369576 0.86 PTGS2 (0.79) PTGS2CDC42RAC1PTGS1PAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0284076-B1 Process for preparing (+)-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds SYNTEX INC (US) 1994-06-08 EP disclosed
EP-0275092-B1 PROCESS FOR PREPARING (+)-1,2-DIHYDRO-3H-PYRROLO(1,2-A)PYRROLE-1,7-DICARBOXYLATES SYNTEX (U.S.A.) INC. (US) 1992-06-03 EP disclosed
EP-0284076-A1 Process for preparing (+)-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds SYNTEX (U.S.A.) INC. (US) 1988-09-28 EP disclosed
EP-0275092-A1 Process for preparing (+)-1,2-dihydro-3H-pyrrolo(1,2-a)pyrrole-1,7-dicarboxylates SYNTEX (U.S.A.) INC. (US) 1988-07-20 EP disclosed
US-4089969-A ANTIINFLAMMATORY, ANALGESIC, ANTIPYRETIC, SMOOTH MUSCLE RELAXANT SYNTEX (U.S.A.) INC. (US) 1978-05-16 US disclosed