SCHEMBL9387643

SCHEMBL9387643

Nc1nc(O)c2c(n1)NC[C@@H](CCc1ccc(C(=O)N[C@H](CCC(=O)O)C(=O)O)o1)C2

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GART P22102 7/20 0.59
DHFR P00374 3/20 0.59
ATIC P31939 4/20 0.46
FOLR2 P14207 1/20 0.46
FOLR1 P15328 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9382833 1.00 GART (0.59) GARTDHFRATICFOLR2FOLR1
SCHEMBL9387634 1.00 GART (0.59) GARTDHFRATICFOLR2FOLR1
SCHEMBL9382816 1.00 GART (0.59) GARTDHFRATICFOLR2FOLR1
SCHEMBL9388635 0.94 DHFR (0.54) GARTDHFRATICFOLR2FOLR1
SCHEMBL9383773 0.94 DHFR (0.54) GARTDHFRATICFOLR2FOLR1
Lometrexol SCHEMBL9045915 0.88 GART (0.75) GARTDHFRATIC
Lometrexol SCHEMBL12022771 0.88 GART (0.75) GARTDHFRATIC
SCHEMBL7487513 0.85 GART (0.71) GARTDHFRATIC
SCHEMBL8820483 0.85 GART (0.60) GARTDHFRATICFOLR2FOLR1
SCHEMBL7488545 0.85 GART (0.71) GARTDHFRATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0343801-B1 N-(5,6,7,8-tetrahydropyrido(2,3-D)pyrimidin-6-yl-alkanoyl)-glutamic acid derivatives UNIV PRINCETON (US) 1994-08-03 EP claimed
US-4882334-A ANTITUMOR AGENTS INHIBIT ENZYMES WHICH USE FOLIC ACID OR ITS METABOLITES AS SUBSTRATE; ANTICARCINOGENIC THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-11-21 US claimed