SCHEMBL9387679

SCHEMBL9387679

O=c1cc(O)c(=O)c2c(Cl)cc(Cl)cc2[nH]1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 3/20 0.50
GRIN3B O60391 3/20 0.50
GRIN1 Q05586 3/20 0.50
GRIN2A Q12879 3/20 0.50
GRIN2B Q13224 3/20 0.50
GRIN2C Q14957 3/20 0.50
GRIN3A Q8TCU5 3/20 0.50
CA12 O43570 1/20 0.49
CA9 Q16790 1/20 0.49
EEF2K O00418 1/20 0.48
PLK4 O00444 1/20 0.48
IKBKB O14920 1/20 0.48
DYRK3 O43781 1/20 0.48
PIM1 P11309 1/20 0.48
CDK2 P24941 1/20 0.48
AKT1 P31749 1/20 0.48
AKT2 P31751 1/20 0.48
CLK2 P49760 1/20 0.48
GSK3B P49841 1/20 0.48
IRAK1 P51617 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6579538 0.89 GRIN2D (0.53) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9393386 0.83 KDM4E (0.41) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9390017 0.81 GRIN2D (0.49) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL28344828 0.80 GRIN2D (0.48) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9389802 0.80 MAPT (0.47) MEN1CYP1A2CYP2C9TSHRCYP2C19
SCHEMBL9389364 0.76 GRIN2D (0.41) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9390079 0.73 KDM4E (0.33) MEN1KMT2AHTTKDM4EALDH1A1
SCHEMBL9388992 0.73 KDM4E (0.42) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL13412891 0.73 CA12 (0.49) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9007833 0.72 GRIN2D (0.59) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994007500-A1 2,5-DIHYDRO-2,5-DIOXO-1H-AZEPINES AND 2,5-DIHYDRO-2-OXO-1H-AZEPINES AND THE USE THEREOF AS EXCITATORY AMINO ACID AND GLYCINE RECEPTOR ANTAGONISTS WEBER ECKARD (US) 1994-04-14 WO disclosed