SCHEMBL9388992

SCHEMBL9388992

Cc1cc2[nH]c(=O)cc(O)c(=O)c2c(Cl)c1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
ERN1 O75460 1/20 0.41
GRIN2D O15399 4/20 0.40
GRIN3B O60391 4/20 0.40
GRIN1 Q05586 4/20 0.40
GRIN2A Q12879 4/20 0.40
GRIN2B Q13224 4/20 0.40
GRIN2C Q14957 4/20 0.40
GRIN3A Q8TCU5 4/20 0.40
TP53 P04637 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
UPP1 Q16831 1/20 0.36
JAK1 P23458 1/20 0.36
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9392576 0.86 KDM4E (0.40) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9390017 0.85 GRIN2D (0.49) KDM4EALDH1A1HPGDERN1GRIN2D
SCHEMBL9392823 0.77 ERN1 (0.41) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9389405 0.76 DAO (0.41) KDM4EALDH1A1GRIN2DGRIN3BGRIN1
SCHEMBL9389364 0.76 GRIN2D (0.41) KDM4EALDH1A1HPGDGRIN2DGRIN3B
SCHEMBL9389273 0.74 GRIN2D (0.47) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9389038 0.74 ERN1 (0.38) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL9387679 0.73 GRIN2D (0.50) KDM4EALDH1A1HPGDGRIN2DGRIN3B
SCHEMBL9389961 0.73 GRIN2D (0.58) ALDH1A1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL9393386 0.71 KDM4E (0.41) KDM4EALDH1A1GRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994007500-A1 2,5-DIHYDRO-2,5-DIOXO-1H-AZEPINES AND 2,5-DIHYDRO-2-OXO-1H-AZEPINES AND THE USE THEREOF AS EXCITATORY AMINO ACID AND GLYCINE RECEPTOR ANTAGONISTS WEBER ECKARD (US) 1994-04-14 WO disclosed