SCHEMBL9389777

SCHEMBL9389777

O=c1[nH]c2ccc(F)cc2c(=O)cc1O

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DAO P14920 6/20 0.65
DDO Q99489 3/20 0.60
KEAP1 Q14145 1/20 0.60
NFE2L2 Q16236 1/20 0.60
KDM4E B2RXH2 4/20 0.54
ALDH1A1 P00352 3/20 0.54
HPGD P15428 2/20 0.54
LMNA P02545 1/20 0.54
FEN1 P39748 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.51
GHSR Q92847 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
HTT P42858 1/20 0.47
PGR P06401 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9007832 0.86 DAO (0.65) DAODDOKDM4EALDH1A1HPGD
SCHEMBL9387730 0.79 HPGD (0.60) DAODDOKDM4EALDH1A1HPGD
SCHEMBL9007825 0.79 DAO (0.65) DAOKDM4EALDH1A1HPGDLMNA
SCHEMBL9387632 0.79 DAO (0.65) DAODDOKDM4EALDH1A1HPGD
SCHEMBL16767846 0.79 DAO (1.00) DAODDOKDM4EALDH1A1HPGD
SCHEMBL9387925 0.79 DAO (0.53) DAODDO
SCHEMBL3422670 0.77 KDM4E (0.53) DAODDOKEAP1NFE2L2KDM4E
SCHEMBL2639080 0.77 DAO (0.61) DAODDOKDM4EALDH1A1HPGD
SCHEMBL9393317 0.76 FASN (0.57) DAODDOMEN1KMT2A
SCHEMBL9393070 0.76 DAO (0.63) DAODDOKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994007500-A1 2,5-DIHYDRO-2,5-DIOXO-1H-AZEPINES AND 2,5-DIHYDRO-2-OXO-1H-AZEPINES AND THE USE THEREOF AS EXCITATORY AMINO ACID AND GLYCINE RECEPTOR ANTAGONISTS WEBER ECKARD (US) 1994-04-14 WO disclosed