SCHEMBL9389927

SCHEMBL9389927

CCc1cc(CC)c2[nH]c(=O)c(O)cc(=O)c2c1CC

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DAO P14920 6/20 0.49
DDO Q99489 3/20 0.42
GRIN1 Q05586 3/20 0.39
GRIN2D O15399 2/20 0.39
GRIN3B O60391 2/20 0.39
GRIN2A Q12879 2/20 0.39
GRIN2B Q13224 2/20 0.39
GRIN2C Q14957 2/20 0.39
GRIN3A Q8TCU5 2/20 0.39
KDM4E B2RXH2 1/20 0.34
PKM P14618 1/20 0.34
PDE2A O00408 1/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE1C Q14123 1/20 0.33
GPR35 Q9HC97 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
PGR P06401 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9389400 0.90 DAO (0.49) DAODDOGRIN1GRIN2DGRIN3B
SCHEMBL9388974 0.85 DAO (0.49) DAODDOGRIN1GRIN2DGRIN3B
SCHEMBL9389013 0.82 DAO (0.58) DAODDOGRIN1GRIN2DGRIN3B
SCHEMBL9389943 0.80 DAO (0.42) DAODDOKDM4EPKMPDE2A
SCHEMBL9389293 0.79 DAO (0.48) DAODDOGRIN1GRIN2DGRIN3B
SCHEMBL9393239 0.79 DAO (0.48) DAODDOGRIN1GRIN2DGRIN3B
SCHEMBL9389908 0.78 DAO (0.50) DAODDOGRIN1GRIN2DGRIN3B
SCHEMBL9390047 0.77 DAO (0.42) DAODDOGRIN1GRIN2AKDM4E
SCHEMBL9393136 0.75 DAO (0.43) DAODDOKDM4EPKMPDE2A
SCHEMBL9387654 0.75 DAO (0.50) DAODDOGRIN1GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994007500-A1 2,5-DIHYDRO-2,5-DIOXO-1H-AZEPINES AND 2,5-DIHYDRO-2-OXO-1H-AZEPINES AND THE USE THEREOF AS EXCITATORY AMINO ACID AND GLYCINE RECEPTOR ANTAGONISTS WEBER ECKARD (US) 1994-04-14 WO disclosed