SCHEMBL9401068

SCHEMBL9401068

COc1ccc(-c2cnc(N3CCN(CCCCN)CC3)nc2)cc1OC

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 6/20 0.55
TLR9 Q9NR96 5/20 0.55
TLR8 Q9NR97 4/20 0.55
MAP4K1 Q92918 3/20 0.50
IL2 P60568 1/20 0.50
DRD2 P14416 8/20 0.46
DRD4 P21917 8/20 0.46
DRD3 P35462 8/20 0.46
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
HTR1A P08908 2/20 0.46
HTR7 P34969 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9401076 0.97 TLR7 (0.56) TLR7TLR9TLR8MAP4K1IL2
SCHEMBL9401042 0.85 HSD17B10 (0.59) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL9401008 0.82 HTR1A (0.62) DRD2DRD3HTR1AHTR7
SCHEMBL9400941 0.81 HSD17B10 (0.64) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL9400948 0.78 SLC6A4 (0.52) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL3196772 0.78 HSD17B10 (0.62) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL9400960 0.78 CYP2D6 (0.54) DRD2DRD4DRD3HTR1A
SCHEMBL9480334 0.77 HTR1A (0.51) TLR7TLR9TLR8DRD2DRD4
Hydrochloric Acid SCHEMBL3188909 0.77 HSD17B10 (0.60) DRD2DRD4DRD3HTR1AHTR7
SCHEMBL7053849 0.74 DRD3 (0.56) DRD2DRD4DRD3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5314884-A Antidepressants, anxiolytic agents TROPONWERKE GMBH & CO. (DE) 1994-05-24 US disclosed
US-5187276-A Anxiolytics, neuroleptics, antidepressants, and nootropic agents TROPONWERKE GMBH & CO. KG. (DE) 1993-02-16 US disclosed
US-4988809-A CENTRAL NERVOUS SYSTEM TROPONWERKE GMBH & CO., KG (DE) 1991-01-29 US disclosed
EP-0129128-B1 2-PYRIMIDINYL-1-PIPERAZINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM Troponwerke GmbH & Co. KG (DE) 1990-11-22 EP disclosed
US-4937343-A NEUROLEPTICS OR ANTIDEPRESSANTS TROPONWERKE GMBH & CO. KG (DE) 1990-06-26 US disclosed
US-4818756-A CENTRAL NERVOUS SYSTEM DISORDERS TROPONWERKE GMBH & CO., KG (DE) 1989-04-04 US disclosed
EP-0129128-A2 2-Pyrimidinyl-1-piperazine derivatives, process for their preparation and medicines containing them Troponwerke GmbH & Co. KG (DE) 1984-12-27 EP disclosed