SCHEMBL9401756

SCHEMBL9401756

COC(=O)C1=C(C)NC(C)=C(C(=O)OCC=Cc2ccc(Cc3ncc[nH]3)cc2)C1c1cccc2ncoc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 15/20 0.43
CYP2C9 P11712 5/20 0.39
CYP1A2 P05177 4/20 0.39
CYP3A4 P08684 4/20 0.39
CYP2C19 P33261 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
NR1I2 O75469 2/20 0.39
ABCB11 O95342 2/20 0.39
NR3C1 P04150 2/20 0.39
ADORA3 P0DMS8 2/20 0.39
CYP2D6 P10635 2/20 0.39
TBXA2R P21731 2/20 0.39
OPRK1 P41145 2/20 0.39
SLC6A3 Q01959 2/20 0.39
PDE4D Q08499 2/20 0.39
SCN5A Q14524 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
MLNR O43193 1/20 0.39
CYP2C8 P10632 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9401598 0.85 CACNA1B (0.47) CACNA1BCYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL9401485 0.85 CACNA1B (0.43) CACNA1BCYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL9401699 0.85 CACNA1B (0.46) CACNA1BCYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL9401549 0.85 CACNA1B (0.47) CACNA1BMEN1KMT2ANR1I2NR3C1
SCHEMBL9401721 0.85 CYP2C9 (0.57) CACNA1BCYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL9401883 0.85 KDM4E (0.55) CACNA1BKMT2AKDM4EHSD17B10ALDH1A1
SCHEMBL9401905 0.85 CACNA1B (0.48) CACNA1BCYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL9401766 0.85 CACNA1B (0.46) CACNA1BCYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL9401885 0.85 CACNA1B (0.46) CACNA1BCYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL7299623 0.84 CACNA1B (0.45) CACNA1BMEN1KMT2ANR1I2NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5286869-A Vasodilators and anticoagulants FUJIREBIO KABUSHIKI KAISHA (JP) 1994-02-15 US disclosed
EP-0403957-A2 Optical active 1,4-dihydropyridine derivates FUJIREBIO INC. (JP) 1990-12-27 EP disclosed