SCHEMBL9401883

SCHEMBL9401883

COC(=O)C1=C(C)NC(C)=C(C(=O)OCC=Cc2ccc(Cc3ncc[nH]3)cc2)C1c1ccco1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.55
POLB P06746 1/20 0.52
CACNA1B Q00975 15/20 0.45
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ADORA2B P29275 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9401771 0.88 CACNA1B (0.48) KDM4ECACNA1BHTTKMT2AHSD17B10
SCHEMBL9401715 0.88 CACNA1B (0.61) CACNA1BHTTKMT2A
SCHEMBL9401726 0.86 CACNA1B (0.60) CACNA1BHTTKMT2AADORA2B
SCHEMBL9401756 0.85 CACNA1B (0.43) KDM4ECACNA1BALDH1A1GAAMAPT
SCHEMBL9401615 0.85 CACNA1B (0.61) CACNA1BHTTKMT2A
SCHEMBL7293440 0.85 CACNA1B (0.64) CACNA1BGAAHTTKMT2A
SCHEMBL9401598 0.85 CACNA1B (0.47) KDM4ECACNA1BALDH1A1GAAMAPT
SCHEMBL9401579 0.84 CACNA1B (0.46) KDM4ECACNA1BHTTKMT2AHSD17B10
SCHEMBL9401766 0.84 CACNA1B (0.46) KDM4ECACNA1BALDH1A1GAAMAPT
SCHEMBL9401521 0.84 MEN1 (0.52) CACNA1BALDH1A1MAPTHTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5286869-A Vasodilators and anticoagulants FUJIREBIO KABUSHIKI KAISHA (JP) 1994-02-15 US disclosed
EP-0403957-A2 Optical active 1,4-dihydropyridine derivates FUJIREBIO INC. (JP) 1990-12-27 EP disclosed