SCHEMBL9402952

SCHEMBL9402952

CC(C)(C)NC(=O)NC(=O)[C@H]1CC[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 7/20 0.68
CYP3A4 P08684 6/20 0.68
ALDH1A1 P00352 4/20 0.68
SMN1; SMN2 Q16637 4/20 0.68
MAPT P10636 4/20 0.68
MAPK1 P28482 4/20 0.68
TSHR P16473 4/20 0.68
SHBG P04278 4/20 0.68
SERPINA6 P08185 4/20 0.68
NR3C1 P04150 4/20 0.68
PGR P06401 4/20 0.68
AR P10275 3/20 0.68
GPBAR1 Q8TDU6 3/20 0.68
SIGMAR1 Q99720 3/20 0.68
CYP2C9 P11712 2/20 0.68
HIF1A Q16665 2/20 0.68
ABCB11 O95342 2/20 0.68
NR1I2 O75469 2/20 0.68
NR3C2 P08235 2/20 0.68
CYP2C19 P33261 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9402961 1.00 LMNA (0.68) LMNACYP3A4ALDH1A1SMN1; SMN2MAPT
SCHEMBL9402966 1.00 LMNA (0.68) LMNACYP3A4ALDH1A1SMN1; SMN2MAPT
SCHEMBL6263255 0.92 LMNA (0.73) LMNACYP3A4ALDH1A1SMN1; SMN2MAPT
SCHEMBL6263252 0.92 LMNA (0.73) LMNACYP3A4ALDH1A1SMN1; SMN2MAPT
SCHEMBL8804072 0.86 LMNA (0.73) LMNACYP3A4ALDH1A1SMN1; SMN2MAPT
SCHEMBL8804080 0.86 LMNA (0.73) LMNACYP3A4ALDH1A1SMN1; SMN2MAPT
SCHEMBL8804068 0.86 LMNA (0.73) LMNACYP3A4ALDH1A1SMN1; SMN2MAPT
SCHEMBL8802536 0.85 LMNA (0.72) LMNACYP3A4ALDH1A1SMN1; SMN2MAPT
SCHEMBL8802547 0.85 LMNA (0.72) LMNACYP3A4ALDH1A1SMN1; SMN2MAPT
SCHEMBL8802540 0.85 LMNA (0.72) LMNACYP3A4ALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5342948-A Antiandrogens; ozonation, amination, reduction of androstane derivative with acyl(urea or thiourea) FARMITALIA CARLO ERBA S.R.L. (IT) 1994-08-30 US disclosed
WO-1993002096-A1 PROCESS FOR THE PREPARATION OF 17β-SUBSTITUTED-4-AZA-5α-ANDROSTAN-3-ONE DERIVATIVES FARMITALIA CARLO ERBA S.R.L. (IT) 1993-02-04 WO disclosed
EP-0523688-A1 Process for the preparation of 17beta-substituted-4-aza-5alpha-androstan-3-one derivatives PHARMACIA S.p.A. (IT) 1993-01-20 EP disclosed