SCHEMBL9403595

SCHEMBL9403595

Nc1c(F)c(N2CC(N)C3(CC3)C2)cc2c1c(=O)c(C(=O)O)cn2C1CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.51
HRH3 Q9Y5N1 1/20 0.51
POLB P06746 2/20 0.49
CACNA1F O60840 1/20 0.49
MAPK1 P28482 1/20 0.49
CACNA1D Q01668 1/20 0.49
CACNA1S Q13698 1/20 0.49
CACNA1C Q13936 1/20 0.49
GSK3B P49841 10/20 0.47
TOP2A P11388 2/20 0.44
TOP2B Q02880 2/20 0.44
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 3/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
LMNA P02545 2/20 0.43
HPGD P15428 2/20 0.43
HSD17B10 Q99714 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9023271 0.99 KCNH2 (0.50) KCNH2HRH3POLBCACNA1FMAPK1
Hydrochloric Acid SCHEMBL9023276 0.99 KCNH2 (0.50) KCNH2HRH3POLBCACNA1FMAPK1
SCHEMBL8775506 0.83 KDM4E (0.64) TOP2ATOP2BALDH1A1KDM4ELMNA
SCHEMBL9023644 0.83 KCNH2 (0.58) KCNH2HRH3POLBCACNA1FMAPK1
SCHEMBL9023635 0.83 KCNH2 (0.58) KCNH2HRH3POLBCACNA1FMAPK1
Hydrochloric Acid SCHEMBL9023258 0.82 KDM4E (0.63) TOP2ATOP2BALDH1A1KDM4ELMNA
Hydrochloric Acid SCHEMBL9023266 0.82 KDM4E (0.63) TOP2ATOP2BALDH1A1KDM4ELMNA
SCHEMBL9079484 0.82 CACNA1F (0.67) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL9080555 0.82 POLB (0.57) KCNH2POLBCACNA1FMAPK1CACNA1D
SCHEMBL9500959 0.81 KCNH2 (0.71) KCNH2HRH3POLBCACNA1FMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-6049060-A None JP disclosed
JP-H0649060-A 5-AMINO-7-@(3754/24)5-AZASPIRO(2,4)HEPTAN-5-YL)QUINOLINE-3-CARBOXYLIC ACID DERIVATIVE HOKURIKU SEIYAKU CO LTD 1994-02-22 JP disclosed
JP-H00649060-A 0001-01-01 JP disclosed