SCHEMBL9408574

SCHEMBL9408574

O=[N+]([O-])C=C1NCC=CN1Cc1ccc(Br)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.46
CHRNA4 P43681 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CHRNA1 P02708 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA7 P36544 1/20 0.43
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPK1 P28482 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CYP19A1 P11511 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9408704 0.88 CHRNB2 (0.49) CHRNB2CHRNA4SMN1; SMN2CHRNA1CHRNA3
SCHEMBL9408592 0.87 CHRNB2 (0.46) CHRNB2CHRNA4SMN1; SMN2CHRNA1CHRNA3
SCHEMBL7993660 0.86 CHRNB2 (0.46) CHRNB2CHRNA4SMN1; SMN2CHRNA1CHRNA3
Hydrochloric Acid SCHEMBL10734635 0.85 CHRNB2 (0.46) CHRNB2CHRNA4SMN1; SMN2CHRNA1CHRNA3
SCHEMBL9068992 0.84 CHRNB2 (0.52) CHRNB2CHRNA4SMN1; SMN2CHRNA1CHRNA3
SCHEMBL10892508 0.84 CHRNB2 (0.43) CHRNB2CHRNA4SMN1; SMN2CHRNA1CHRNA3
Hydrochloric Acid SCHEMBL10483929 0.83 CHRNB2 (0.51) CHRNB2CHRNA4SMN1; SMN2CHRNA1CHRNA3
SCHEMBL9408581 0.82 SMN1; SMN2 (0.47) CHRNB2CHRNA4SMN1; SMN2CHRNA1CHRNA3
SCHEMBL1019754 0.82 CHRNB2 (0.70) CHRNB2CHRNA4SMN1; SMN2CHRNA1CHRNA3
Hydrochloric Acid SCHEMBL10483913 0.81 CHRNB2 (0.69) CHRNB2CHRNA4SMN1; SMN2CHRNA1CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4590272-A INSECTICIDES, MITICIDES, NEMATOCIDES NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1986-05-20 US claimed
EP-0623601-A1 N-(3-Fluorobenzyl)heterocyclic derivatives and their use as pesticides SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1994-11-09 EP disclosed