SCHEMBL9409583

SCHEMBL9409583

COC(=O)c1ccc(C2CNC(=O)C2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.57
PDE4A P27815 10/20 0.55
PDE4B Q07343 5/20 0.55
PDE4C Q08493 5/20 0.55
PDE4D Q08499 5/20 0.55
TSHR P16473 3/20 0.55
PKM P14618 1/20 0.48
MAPK1 P28482 2/20 0.47
TP53 P04637 1/20 0.47
GAA P10253 2/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
GLA P06280 1/20 0.47
HPGD P15428 1/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
ATM Q13315 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CYP3A4 P08684 2/20 0.46
VEGFA P15692 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7233581 0.84 HTT (0.52) HTTTSHRMAPK1TP53GAA
SCHEMBL31115506 0.84 PDE4A (0.52) HTTPDE4APDE4BPDE4CPDE4D
SCHEMBL19780858 0.83 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL19202429 0.79 HTT (0.56) HTTTSHRMAPK1TP53GAA
SCHEMBL15239841 0.79 KDM4E (0.53) HTTTSHRMAPK1GAAKDM4E
Acetic Acid Methyl Ester SCHEMBL28100313 0.79 PDE4A (0.51) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL18117753 0.78 TSHR (0.69) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL1268717 0.78 TSHR (0.69) PDE4APDE4BPDE4CPDE4DTSHR
Hydrochloric Acid SCHEMBL15240346 0.78 KDM4E (0.51) HTTTSHRMAPK1GAAKDM4E
SCHEMBL13267179 0.77 ALDH1A1 (0.55) HTTTSHRGAAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0604800-A1 4- 4- 4-(carboxyalkyl)-phenyl amino carbonyl -phenyl -piperedines as aggregation inhibitors Dr. Karl Thomae GmbH (DE) 1994-07-06 EP disclosed