Anecortave Acetate

Anecortave Acetate

SCHEMBL94110

CC(=O)OCC(=O)[C@@]1(O)CC[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)C3=CC[C@@]21C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 3/20 1.00
FNTA P49354 6/20 0.59
FNTB P49356 6/20 0.59
AR P10275 3/20 0.59
KMT2A Q03164 2/20 0.59
MEN1 O00255 1/20 0.59
BLM P54132 1/20 0.59
TSHR P16473 1/20 0.59
HIF1A Q16665 7/20 0.57
PGR P06401 4/20 0.57
HRH1 P35367 1/20 0.57
LMNA P02545 2/20 0.56
SERPINA6 P08185 1/20 0.56
CHRM1 P11229 1/20 0.56
CYP19A1 P11511 1/20 0.53
CYP3A4 P08684 2/20 0.48
POLB P06746 1/20 0.48
ALDH1A1 P00352 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Anecortave Acetate SCHEMBL8470303 1.00 NR3C1 (1.00) NR3C1FNTAFNTBARKMT2A
Anecortave Acetate SCHEMBL2118233 1.00 NR3C1 (1.00) NR3C1FNTAFNTBARKMT2A
Anecortave Acetate SCHEMBL14612532 1.00 NR3C1 (1.00) NR3C1FNTAFNTBARKMT2A
Anecortave Acetate SCHEMBL8472390 0.96 NR3C1 (0.93) NR3C1FNTAFNTBARKMT2A
SCHEMBL25177986 0.92 NR3C1 (0.85) NR3C1FNTAFNTBARKMT2A
SCHEMBL25184624 0.92 NR3C1 (0.85) NR3C1FNTAFNTBARKMT2A
SCHEMBL23974865 0.92 NR3C1 (0.84) NR3C1FNTAFNTBARKMT2A
SCHEMBL25181307 0.91 NR3C1 (0.83) NR3C1FNTAFNTBARKMT2A
SCHEMBL3437593 0.91 NR3C1 (0.83) NR3C1FNTAFNTBARKMT2A
SCHEMBL3437604 0.90 NR3C1 (0.82) NR3C1FNTAFNTBARKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 8240 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4724079-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION Stealth BioTherapeutics Inc. (US) 2026-04-15 EP claimed
US-20260048096-A1 METHODS AND COMPOSITIONS FOR PRESERVING THE RETINAL OUTER NUCLEAR LAYER (ONL), PHOTORECEPTORS, AND RETINAL THICKNESS STEALTH BIOTHERAPEUTICS INC. (US) 2026-02-19 US claimed
EP-4596049-A2 PEPTIDE FOR USE IN PREVENTING OR TREATING MACULAR DEGENERATION Stealth BioTherapeutics Inc. (US) 2025-08-06 EP claimed
EP-4302829-B1 PEPTIDE FOR USE IN PREVENTING OR TREATING MACULAR DEGENERATION STEALTH BIOTHERAPEUTICS INC (US) 2025-05-21 EP claimed
US-12268779-B2 Ophthalmic emulsion ALCON INC. (CH) 2025-04-08 US claimed
US-20250108001-A1 TOPICAL OCULAR ADMINISTRATION OF AMBROXOL FOR OCULAR PAIN NEUVISION DEVELOPMENT LLC 2025-04-03 US claimed
US-20250090621-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION STEALTH BIOTHERAPEUTICS INC. (US) 2025-03-20 US claimed
US-20250057962-A1 PROCESSABLE COMPOSITIONS AND USE FOR THE SAME RIPPLE THERAPEUTICS CORPORATION (CA) 2025-02-20 US claimed
CN-118994021-B Method for recovering imidazole from anecortave acetate byproduct imidazole hydrochloride 山东同新药业有限公司 2025-02-07 CN claimed
CN-119317415-A Topical ocular administration of ambroxol for ocular pain 纽视发展有限责任公司 2025-01-14 CN claimed
US-5679666-A ADMINISTERING TOPICALLY, SYSTEMICALLY OR INTRAOCULARLY TO A HOST STEROIDS SELECTED FROM PREGNADIEN DERIVATIVES, HYDROXYPROGESTERONE AND TETRAHYDROCORTEXOLONE ALCON LABORATORIES, INC. (US) 1997-10-21 US claimed
US-5371078-A Angiostatic steroids and methods and compositions for controlling ocular hypertension ALCON LABORATORIES, INC. (US) 1994-12-06 US claimed
EP-0614463-A1 ANGIOSTATIC STEROIDS ALCON LABORATORIES, INC. (US) 1994-09-14 EP claimed
WO-1993010141-A2 ANGIOSTATIC STEROIDS ALCON LABORATORIES, INC. (US) 1993-05-27 WO claimed
US-4749649-A Microbial Δ1-dehydrogenation process using a scavenger of toxic oxygen THE UPJOHN COMPANY (US) 1988-06-07 US claimed
US-4684610-A ARTHROBACTER OR BACTERIUM THE UPJOHN COMPANY (US) 1987-08-04 US claimed
EP-0127294-B1 STEROID DEHYDROGENATION THE UPJOHN COMPANY (US) 1986-12-17 EP claimed
EP-0127294-A1 Steroid dehydrogenation THE UPJOHN COMPANY (US) 1984-12-05 EP claimed
US-4154748-A Phosphate catalyzed acylation of steroidal tertiary alcohols THE UPJOHN COMPANY (US) 1979-05-15 US claimed
US-4041055-A SULFENYLATION, MICHAEL ADDITION, REACTION WITH THIOPHILE, HYDROLYSIS THE UPJOHN COMPANY (US) 1977-08-09 US claimed