SCHEMBL9412931

SCHEMBL9412931

COc1cc(N)c(Cl)cc1C(=O)N[C@H]1C[C@H]2COC[C@@H](C1)N2Cc1ccc(F)cc1

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.69
HTR4 Q13639 4/20 0.61
DRD3 P35462 3/20 0.56
DRD4 P21917 4/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
ADRA2A P08913 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
ADRA2B P18089 1/20 0.56
ADRA2C P18825 1/20 0.56
ACHE P22303 1/20 0.56
SLC6A2 P23975 1/20 0.56
HTR2A P28223 1/20 0.56
HTR2C P28335 1/20 0.56
ADRA1A P35348 1/20 0.56
OPRK1 P41145 1/20 0.56
HTR2B P41595 1/20 0.56
CHRNA4 P43681 1/20 0.56
HTR3A P46098 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9412933 1.00 DRD2 (0.69) DRD2HTR4DRD3DRD4CYP1A2
SCHEMBL11237366 0.93 DRD2 (0.71) DRD2HTR4DRD3DRD4CYP1A2
SCHEMBL11237369 0.93 DRD2 (0.71) DRD2HTR4DRD3DRD4CYP1A2
SCHEMBL9412905 0.92 DRD2 (0.70) DRD2HTR4DRD3DRD4CYP1A2
SCHEMBL11232514 0.92 DRD2 (0.70) DRD2HTR4DRD3DRD4CYP1A2
SCHEMBL9412901 0.92 DRD2 (0.70) DRD2HTR4DRD3DRD4CYP1A2
SCHEMBL11232518 0.92 DRD2 (0.70) DRD2HTR4DRD3DRD4CYP1A2
SCHEMBL9413082 0.91 DRD2 (0.58) DRD2HTR4DRD3DRD4CYP1A2
SCHEMBL9413072 0.91 DRD2 (0.58) DRD2HTR4DRD3DRD4CYP1A2
SCHEMBL11227150 0.91 DRD2 (0.69) DRD2HTR4DRD3DRD4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623621-A1 Oxazabicyclo derivatives and their use as 5-HT4 receptor agonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1994-11-09 EP disclosed