SCHEMBL9416630

SCHEMBL9416630

COc1ccc(CN(C)Cc2ccc(O)c(OC)c2)cc1O

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.57
NFKB1 P19838 2/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
LMNA P02545 2/20 0.55
APEX1 P27695 1/20 0.55
TAAR1 Q96RJ0 2/20 0.54
MAPK1 P28482 1/20 0.54
TUBB4A P04350 2/20 0.54
TUBB P07437 2/20 0.54
TUBA3C P0DPH7 2/20 0.54
TUBA1B P68363 2/20 0.54
TUBA4A P68366 2/20 0.54
TUBB4B P68371 2/20 0.54
TUBB3 Q13509 2/20 0.54
TUBB2A Q13885 2/20 0.54
TUBB8 Q3ZCM7 2/20 0.54
TUBA3E Q6PEY2 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11648537 0.83 TAAR1 (0.61) TSHRNFKB1CYP3A4LMNATAAR1
SCHEMBL30873093 0.83 TUBB4A (0.75) TSHRNFKB1CYP1A2CYP3A4MEN1
SCHEMBL27183302 0.83 TUBB4A (0.75) TSHRNFKB1CYP1A2CYP3A4MEN1
SCHEMBL15042812 0.83 TUBB4A (0.75) TSHRNFKB1CYP1A2CYP3A4MEN1
SCHEMBL29442255 0.83 TUBB4A (0.75) TSHRNFKB1CYP1A2CYP3A4MEN1
SCHEMBL3691695 0.83 CYP1A2 (0.59) TSHRNFKB1CYP1A2CYP3A4MEN1
SCHEMBL9416555 0.82 TSHR (0.54) TSHRNFKB1CYP1A2CYP3A4MEN1
SCHEMBL27777910 0.81 TSHR (0.62) TSHRNFKB1CYP1A2CYP3A4MEN1
SCHEMBL10049174 0.80 CYP1A2 (0.60) TSHRNFKB1CYP1A2CYP3A4MEN1
SCHEMBL13131818 0.80 TAAR1 (0.61) TSHRNFKB1CYP3A4LMNATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0613879-A1 PHELLODENDRINE ANALOGS AND ALLERGY TYPE IV SUPPRESSOR CONTAINING THE SAME AS ACTIVE INGREDIENT TSUMURA & CO. (JP) 1994-09-07 EP disclosed