SCHEMBL9417868

SCHEMBL9417868

CCc1cc(C(=O)CCCCC(=O)O)c(OC)cc1OC

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.45
POLB P06746 2/20 0.41
MAPK1 P28482 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
STING1 Q86WV6 2/20 0.40
CYP3A4 P08684 2/20 0.40
HTR4 Q13639 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC1 Q13547 1/20 0.40
KMT2A Q03164 1/20 0.40
HTT P42858 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9417829 0.87 HMGCR (0.54) PDE4BCYP3A4KMT2AHTT
SCHEMBL8893882 0.80 HMGCR (0.56) STING1CYP3A4KMT2AHTTTAAR1
SCHEMBL8902437 0.79 KDM4E (0.53) MAPK1CYP3A4KMT2ATAAR1
SCHEMBL14525269 0.78 TAAR1 (0.51) STING1CYP3A4KMT2ATAAR1
SCHEMBL14525270 0.78 HPGDS (0.47) STING1CYP3A4KMT2ATAAR1
SCHEMBL31113388 0.77 HTT (0.53) STING1CYP3A4KMT2AHTT
SCHEMBL7261534 0.76 PDE4B (0.60) PDE4BMAPK1KMT2AHTT
SCHEMBL8824020 0.75 HMGCR (0.54) PDE4BPOLBMAPK1SMN1; SMN2CYP3A4
SCHEMBL11836438 0.75 STING1 (0.57) STING1HTR4HTT
SCHEMBL14925385 0.75 TSHR (0.54) PDE4BSMN1; SMN2HDAC8HDAC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5294613-A Benzene derivatives of p-substituted ether and acid or ester ELI LILLY AND COMPANY (US) 1994-03-15 US disclosed
US-5098613-A Aromatic ethers for treatment of mammals ELI LILLY AND COMPANY (US) 1992-03-24 US disclosed
US-4945099-A LEUKOTRIENE ANTAGONIST ELI LILLY AND COMPANY (US) 1990-07-31 US disclosed
EP-0276065-B1 ANTI-INFLAMMATORY AGENTS ELI LILLY AND COMPANY (US) 1990-06-06 EP disclosed
EP-0276065-A1 Anti-inflammatory agents ELI LILLY AND COMPANY (US) 1988-07-27 EP disclosed