SCHEMBL9419243

SCHEMBL9419243

COc1ccc(-c2ccc(C(=O)O)c(F)c2F)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.64
CYP2C19 P33261 2/20 0.52
APP P05067 1/20 0.52
PRKAB2 O43741 3/20 0.52
PRKAG1 P54619 3/20 0.52
PRKAA2 P54646 3/20 0.52
PRKAA1 Q13131 3/20 0.52
PRKAG3 Q9UGI9 3/20 0.52
PRKAG2 Q9UGJ0 3/20 0.52
PRKAB1 Q9Y478 3/20 0.52
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 2/20 0.50
GAA P10253 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
POLB P06746 1/20 0.47
HPGD P15428 1/20 0.47
CA1 P00915 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28188901 0.89 SMN1; SMN2 (0.62) SMN1; SMN2CYP2C19APPPRKAB2PRKAG1
SCHEMBL18873501 0.84 HSD17B10 (0.53) SMN1; SMN2CYP2C19KDM4EALDH1A1GAA
SCHEMBL22561016 0.82 CA12 (0.52) SMN1; SMN2CYP2C19APPKDM4ECYP1A2
SCHEMBL9419340 0.81 SMN1; SMN2 (0.47) SMN1; SMN2PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL505335 0.81 KDM4E (0.50) CYP2C19APPKDM4EALDH1A1CYP2C9
SCHEMBL9419305 0.81 RARB (0.53) SMN1; SMN2PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL12822797 0.81 CYP2C19 (0.51) SMN1; SMN2CYP2C19APPPRKAB2PRKAG1
SCHEMBL30585141 0.80 BCL2L1 (0.52) KDM4EALDH1A1CYP2C9HPGDCA1
SCHEMBL5571280 0.80 HSD17B10 (0.59) SMN1; SMN2CYP2C19APPKDM4EALDH1A1
SCHEMBL26639280 0.80 BCL2L1 (0.52) KDM4EALDH1A1CYP2C9HPGDCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0363458-B1 2,3-DIFLUOROBENZENES MERCK PATENT GMBH (DE) 1994-08-03 EP disclosed
US-5087764-A Deprotonation of a 1-substituted-2,3-difluorobenzene using an organometallic compound and reacting the reaction product with an electrophile Merck Patent Gesellschaft mit beschrankter Hafung (DE) 1992-02-11 US disclosed