SCHEMBL9424313

SCHEMBL9424313

CCCCc1nc2cccc(C)n2c(=O)c1Cc1ccc(I)cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 4/20 0.40
CCR5 P51681 1/20 0.40
HTT P42858 1/20 0.40
MAPT P10636 1/20 0.37
APLNR P35414 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
AGTR1 P30556 1/20 0.36
AGTR2 P50052 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11361275 0.77 HTT (0.57) HTTMAPTKDM4EALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL11360548 0.76 HTT (0.56) HTTMAPTKDM4EALDH1A1CYP1A2
SCHEMBL9423837 0.72 MAPT (0.38) HTTMAPTKDM4EALDH1A1POLB
Hydrochloric Acid SCHEMBL11364612 0.71 HTT (0.54) HTTMAPTKDM4EALDH1A1CYP1A2
SCHEMBL11464701 0.71 KDM4E (0.56) HTTMAPTKDM4EALDH1A1POLB
SCHEMBL9424129 0.71 TLR8 (0.34) CCR2CCR5
SCHEMBL11363269 0.70 HTT (0.59) HTTMAPTKDM4EALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL11365039 0.70 KDM4E (0.55) HTTMAPTKDM4EALDH1A1POLB
Hydrochloric Acid SCHEMBL11369573 0.69 HTT (0.57) HTTMAPTKDM4EALDH1A1CYP1A2
SCHEMBL9423387 0.69 HPGD (0.35) CCR2CCR5KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5324729-A Hypotensive agents MERCK & CO., INC. (US) 1994-06-28 US disclosed
US-5166206-A Hypotensive agents, central nervous system disorders, glaucoma or angiotensin antagonist MERCK & CO., INC. (US) 1992-11-24 US disclosed
WO-1991015209-A1 SUBSTITUTED PYRIMIDINES, PYRIMIDINONES AND PYRIDOPYRIMIDINES MERCK & CO., INC. (US) 1991-10-17 WO disclosed