SCHEMBL9424845

SCHEMBL9424845

CC1(C)Oc2ccc([N+](=O)[O-])cc2O1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
TSHR P16473 5/20 0.48
TDP1 Q9NUW8 4/20 0.47
ALDH1A1 P00352 4/20 0.47
CYP3A4 P08684 3/20 0.44
LMNA P02545 1/20 0.43
AKR1B1 P15121 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA9 Q16790 1/20 0.42
HSD17B10 Q99714 2/20 0.42
MEN1 O00255 2/20 0.42
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
ACHE P22303 2/20 0.42
PTPRC P08575 1/20 0.41
S100A4 P26447 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9230962 0.83 ALDH1A1 (0.43) TSHRTDP1ALDH1A1CYP3A4LMNA
SCHEMBL30330229 0.83 ALDH1A1 (0.43) TSHRTDP1ALDH1A1CYP3A4LMNA
SCHEMBL22058720 0.83 CA1 (0.46) TSHRTDP1ALDH1A1CYP3A4LMNA
SCHEMBL10920807 0.83 HSD17B10 (0.46) TSHRTDP1ALDH1A1CYP3A4LMNA
SCHEMBL30849385 0.83 ALDH1A1 (0.43) TSHRTDP1ALDH1A1CYP3A4LMNA
SCHEMBL24179080 0.83 TSHR (0.42) TSHRTDP1ALDH1A1CYP3A4LMNA
SCHEMBL9427783 0.82 AKR1B1 (0.42) CYP1A2CYP2C9CYP2C19TSHRTDP1
SCHEMBL1749524 0.82 MAPT (0.51) CYP1A2CYP2C9CYP2C19TSHRTDP1
SCHEMBL28882693 0.82 HTT (0.44) CYP1A2CYP2C9CYP2C19TSHRTDP1
SCHEMBL12483210 0.82 HTT (0.44) CYP1A2CYP2C9CYP2C19TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019178547-A1 BENZOXAZINE POLYMERS AND METHODS OF MAKING AND USING THE SAME THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-09-19 WO disclosed
US-5318963-A Heterocyclic hydrazide derivatives of monocyclic β-lactam antibiotics E. R. SQUIBB & SONS, INC. (US) 1994-06-07 US disclosed
EP-0525877-A1 Pesticidal heterocyclic compounds SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1993-02-03 EP disclosed
US-5037983-A 6,7-dihydroxyquinoxalines as intermediates to beta-lactam antibiotics E. R. SQUIBB & SONS, INC. (US) 1991-08-06 US disclosed
EP-0420069-A2 Heterocyclic hydrazide derivatives of monocyclic beta-lactam antibiotics E.R. SQUIBB & SONS, INC. (US) 1991-04-03 EP disclosed
EP-0342423-A2 Heteroaroylhydrazide derivatives of monocyclic beta-lactam antibiotics E.R. SQUIBB & SONS, INC. (US) 1989-11-23 EP disclosed
US-4599347-A ANTIULCER AGENTS HOFFMANN-LA ROCHE INC. (US) 1986-07-08 US disclosed
US-4554280-A ANTISECRETORY AGENTS, ANTIULCER AGENTS HOFFMANN-LA ROCHE INC. (US) 1985-11-19 US disclosed
US-4435406-A 2-PYRIDYL DERIVATIVES OF 1,3-DIOXOLO(4,5-F)BENZIMIDAZOLE RING COMPOUNDS HOFFMANN-LA ROCHE INC. (US) 1984-03-06 US disclosed
US-4144341-A ANTIPYRETICS, ANALGESICS AND ANTIINFLAMMATORY AGENTS MERCK & CO., INC. (US) 1979-03-13 US disclosed
US-4000286-A ANALGESICS, ANTIINFLAMMATORY AND ANTIPYRETIC AGENTS MERCK & CO., INC. (US) 1976-12-28 US disclosed