SCHEMBL9425528

SCHEMBL9425528

N#Cc1cc(Br)cc(-n2ccnc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.43
CYP17A1 P05093 1/20 0.43
CYP21A2 P08686 1/20 0.43
CYP3A4 P08684 7/20 0.41
CYP1A2 P05177 5/20 0.41
CYP2C19 P33261 5/20 0.41
CYP2D6 P10635 4/20 0.41
CYP2C9 P11712 2/20 0.41
GAA P10253 1/20 0.41
CYP19A1 P11511 2/20 0.40
ALOX15 P16050 4/20 0.39
HSD17B10 Q99714 3/20 0.39
MAPK1 P28482 2/20 0.39
ALDH1A1 P00352 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 1/20 0.39
ENPP2 Q13822 1/20 0.39
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22745375 0.88 CYP3A4 (0.47) CYP11B1CYP3A4CYP1A2CYP2C19CYP2D6
SCHEMBL6213351 0.86 CYP17A1 (0.39) CYP11B1CYP17A1CYP21A2CYP3A4CYP1A2
SCHEMBL8331340 0.82 CYP11B1 (0.53) CYP11B1CYP17A1CYP21A2CYP3A4CYP19A1
SCHEMBL5224027 0.82 CYP11B1 (0.53) CYP11B1CYP17A1CYP21A2CYP3A4CYP19A1
SCHEMBL5228601 0.81 CYP3A4 (0.41) CYP11B1CYP3A4CYP1A2CYP2C19CYP2D6
SCHEMBL25159951 0.77 ENPP2 (0.39) CYP11B1CYP17A1CYP21A2CYP3A4CYP1A2
SCHEMBL9426009 0.77 CYP3A4 (0.39) CYP11B1CYP3A4CYP1A2CYP2C19CYP2D6
SCHEMBL3531362 0.77 CYP19A1 (0.46) CYP11B1CYP3A4CYP1A2CYP2C19CYP2D6
SCHEMBL3832736 0.75 IDO1 (0.58) CYP11B1CYP3A4CYP1A2CYP2C19CYP2D6
SCHEMBL31420979 0.75 IDO1 (0.58) CYP11B1CYP3A4CYP1A2CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023061263-A1 SHP2 INHIBITOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND USE THEREOF 北京泰德制药股份有限公司 2023-04-20 WO disclosed
US-5276149-A Antibiotics MERCK & CO., INC. (US) 1994-01-04 US disclosed
EP-0538017-A1 2-(N-Imidazoliumphenyl)-carbapenems MERCK & CO. INC. (US) 1993-04-21 EP disclosed