SCHEMBL9427588

SCHEMBL9427588

COc1cc2c(cc1OC)CC(=O)N(CCCN(C)CCC1Cc3cc(OC)c(OC)cc3C1)CC2

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCN4 Q9Y3Q4 3/20 0.68
SLC6A4 P31645 2/20 0.68
CHRM2 P08172 1/20 0.68
HTR1A P08908 1/20 0.68
DRD3 P35462 1/20 0.68
KCNH2 Q12809 1/20 0.68
MAPT P10636 1/20 0.67
CYP3A4 P08684 1/20 0.66
ALOX15 P16050 1/20 0.66
GAA P10253 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
KCNN2 Q9H2S1 4/20 0.38
KCNN3 Q9UGI6 4/20 0.38
KCNN1 Q92952 2/20 0.38
DRD1 P21728 1/20 0.38
DRD4 P21917 1/20 0.38
DRD5 P21918 1/20 0.38
ABCB1 P08183 1/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9427543 0.96 HCN4 (0.64) HCN4SLC6A4CHRM2HTR1ADRD3
SCHEMBL9427426 0.90 HCN4 (0.76) HCN4SLC6A4CHRM2HTR1ADRD3
SCHEMBL9427641 0.87 HCN4 (0.83) HCN4SLC6A4CHRM2HTR1ADRD3
SCHEMBL10846943 0.84 HCN4 (0.72) HCN4SLC6A4CHRM2HTR1ADRD3
SCHEMBL12319782 0.84 HCN4 (0.71) HCN4SLC6A4CHRM2HTR1ADRD3
SCHEMBL10851789 0.82 HCN4 (0.64) HCN4SLC6A4CHRM2HTR1ADRD3
Hydrochloric Acid SCHEMBL10848530 0.81 HCN4 (0.63) HCN4SLC6A4CHRM2HTR1ADRD3
Ivabradine SCHEMBL5163239 0.81 HCN4 (1.00) HCN4SLC6A4CHRM2HTR1ADRD3
Ivabradine SCHEMBL333201 0.81 HCN4 (1.00) HCN4SLC6A4CHRM2HTR1ADRD3
Ivabradine SCHEMBL23472 0.81 HCN4 (1.00) HCN4SLC6A4CHRM2HTR1ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296482-A (Benzocycloalkyl) alkylamines ADIR ET COMPAGNIE (FR) 1994-03-22 US disclosed