SCHEMBL9428433

SCHEMBL9428433

COc1cccc(CCCN(CCO)CCNc2cc(=O)n(C)c(=O)n2C)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 2/20 0.64
SLC6A4 P31645 2/20 0.64
SLC22A2 O15244 1/20 0.64
KCNH2 Q12809 1/20 0.64
SLC47A2 Q86VL8 1/20 0.64
SLC47A1 Q96FL8 1/20 0.64
TAAR1 Q96RJ0 1/20 0.48
CYP1A2 P05177 1/20 0.44
MTNR1A P48039 2/20 0.43
MTNR1B P49286 2/20 0.43
PCSK9 Q8NBP7 2/20 0.43
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MAPT P10636 2/20 0.42
MAPK1 P28482 2/20 0.42
LMNA P02545 1/20 0.42
ADRB2 P07550 1/20 0.42
CYP3A4 P08684 1/20 0.42
HTR1A P08908 1/20 0.42
ADRA2A P08913 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9429589 0.87 ADRB1 (0.75) ADRB1SLC6A4SLC22A2KCNH2SLC47A2
Oxalic Acid SCHEMBL9428952 0.84 SLC22A2 (0.71) ADRB1SLC6A4SLC22A2KCNH2SLC47A2
SCHEMBL9428809 0.84 ADRB1 (0.71) ADRB1SLC6A4SLC22A2KCNH2SLC47A2
SCHEMBL9428818 0.83 ADRB1 (0.64) ADRB1SLC6A4SLC22A2KCNH2SLC47A2
SCHEMBL9428984 0.82 ADRB1 (0.62) ADRB1SLC6A4SLC22A2KCNH2SLC47A2
SCHEMBL9428370 0.81 ADRB1 (0.75) ADRB1SLC6A4SLC22A2KCNH2SLC47A2
SCHEMBL9428374 0.81 ADRB1 (0.75) ADRB1SLC6A4SLC22A2KCNH2SLC47A2
SCHEMBL9428875 0.80 ADRB1 (0.65) ADRB1SLC6A4SLC22A2KCNH2SLC47A2
SCHEMBL9428826 0.79 ADRB1 (0.63) ADRB1SLC6A4SLC22A2KCNH2SLC47A2
Nifekalant SCHEMBL157527 0.78 KCNH2 (1.00) ADRB1SLC6A4SLC22A2KCNH2SLC47A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed