SCHEMBL9429147

SCHEMBL9429147

CCCN(CCNCc1ccc(C#N)cc1)c1cc(=O)n(C)c(=O)n1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 1/20 0.38
CRHR1 P34998 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA4 P22748 1/20 0.37
CA9 Q16790 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.36
MAPK1 P28482 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
IDH1 O75874 1/20 0.34
CACNA1B Q00975 2/20 0.33
CYP1A2 P05177 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
CACNA1G O43497 1/20 0.33
DRD4 P21917 1/20 0.32
RORC P51449 1/20 0.32
NOS3 P29474 2/20 0.32
NOS1 P29475 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9386429 0.82 CHRM2 (0.46) CA12CA1CA2CA4MAPK1
SCHEMBL9385760 0.72 KCNH2 (0.52) SMN1; SMN2
SCHEMBL9429721 0.71 GRIN1 (0.46) HPGDSMN1; SMN2POLB
SCHEMBL2207581 0.70 SCN8A (0.51) SCN8ACA12CA1CA2CA4
SCHEMBL2201948 0.69 SCN8A (0.50) SCN8ACA12CA1CA2CA4
Hydrochloric Acid SCHEMBL2199547 0.69 SCN8A (0.50) SCN8ACA12CA1CA2CA4
SCHEMBL2828109 0.69 SCN8A (0.58) SCN8ACA12CA1CA2CA4
SCHEMBL15831741 0.69 LOXL2 (0.62) SCN8ACA12CA1CA2CA4
SCHEMBL6764095 0.68 SCN8A (0.55) SCN8ACA12CA1CA2CA4
Hydrochloric Acid SCHEMBL2205193 0.68 SCN8A (0.49) SCN8ACA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed
EP-0454498-A2 Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-10-30 EP disclosed