SCHEMBL9433360

SCHEMBL9433360

Cc1ccc(C(=O)C(Br)n2cncn2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.63
HSP90AA1 P07900 1/20 0.63
ALDH1A1 P00352 4/20 0.42
NPSR1 Q6W5P4 2/20 0.42
MEN1 O00255 1/20 0.42
CYP26A1 O43174 2/20 0.41
CYP19A1 P11511 3/20 0.40
PDE4B Q07343 1/20 0.40
CHRM2 P08172 1/20 0.38
ADRA2B P18089 1/20 0.38
DRD3 P35462 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
LMNA P02545 2/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9199550 0.83 KMT2A (0.64) KMT2AHSP90AA1ALDH1A1NPSR1MEN1
SCHEMBL11145904 0.77 HSP90AA1 (0.41) KMT2AHSP90AA1CYP26A1CYP19A1CYP1A2
Bromide SCHEMBL5880713 0.71 GSK3B (0.57) CYP19A1CYP3A4CYP2C19
SCHEMBL11148526 0.70 MAPT (0.36) KMT2AHSP90AA1CYP26A1CYP19A1CYP1A2
SCHEMBL6227295 0.70 CYP19A1 (0.51) KMT2AHSP90AA1ALDH1A1MEN1CYP26A1
SCHEMBL10712303 0.70 HSP90AA1 (0.46) KMT2AHSP90AA1CYP26A1CYP19A1CYP1A2
SCHEMBL10361474 0.70 HSP90AA1 (0.49) KMT2AHSP90AA1CYP26A1CYP19A1PDE4B
SCHEMBL10709431 0.70 HSP90AA1 (0.49) KMT2AHSP90AA1ALDH1A1CYP26A1CYP19A1
SCHEMBL9841086 0.69 MAPT (0.51) KMT2AHSP90AA1MEN1CYP26A1CYP19A1
SCHEMBL9795396 0.69 CYP19A1 (0.49) KMT2AHSP90AA1ALDH1A1NPSR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332753-A Thiazole derivatives, their preparation and their use as fungicides SHELL RESEARCH LIMITED (GB) 1994-07-26 US disclosed
EP-0411718-A2 Thiazole derivatives, their preparation and their use as fungicides SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1991-02-06 EP disclosed