SCHEMBL9433809

SCHEMBL9433809

C=CC(=O)Cc1cnccc1-c1cc(Cl)cc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 5/20 0.36
KCNA5 P22460 2/20 0.35
CTSA P10619 1/20 0.35
GALR3 O60755 1/20 0.34
NR2F2 P24468 1/20 0.34
CYP17A1 P05093 1/20 0.34
CCNC P24863 2/20 0.33
CDK8 P49336 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
MMP13 P45452 1/20 0.33
ROCK2 O75116 1/20 0.32
IDO1 P14902 1/20 0.32
RPS6KA3 P51812 1/20 0.32
WDR5 P61964 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9433930 0.84 GPBAR1 (0.36) GPBAR1KCNA5CCNCCDK8ALDH1A1
SCHEMBL9434105 0.81 RECQL (0.36) KMT2AALDH1A1ROCK2
SCHEMBL9433838 0.81 RPS6KA3 (0.50) GPBAR1CCNCCDK8KMT2AMAPT
SCHEMBL9433530 0.80 RPS6KA3 (0.35) GPBAR1CCNCCDK8MAPTMMP13
SCHEMBL9433512 0.80 SLC22A12 (0.41) GPBAR1CCNCCDK8ALDH1A1MMP13
SCHEMBL9434027 0.80 SLC22A12 (0.40) CDK8ALDH1A1LMNAMAPTMMP13
SCHEMBL9434756 0.79 CYP3A4 (0.39) GPBAR1CYP17A1
SCHEMBL9433807 0.78 LIMK1 (0.41) GPBAR1
SCHEMBL9434449 0.78 RPS6KA3 (0.46) GPBAR1CYP17A1MMP13ROCK2IDO1
SCHEMBL9433871 0.78 PDE4A (0.37) GPBAR1KCNA5CTSACCNCCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed