SCHEMBL9433871

SCHEMBL9433871

C=CC(=O)Cc1cnccc1-c1cccc(I)c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.37
JAK3 P52333 1/20 0.34
GPBAR1 Q8TDU6 5/20 0.34
MMP13 P45452 1/20 0.33
PLCG1 P19174 1/20 0.33
GRK2 P25098 1/20 0.32
CCNC P24863 1/20 0.32
CDK8 P49336 1/20 0.32
FFAR1 O14842 1/20 0.32
ROCK2 O75116 1/20 0.32
MAPT P10636 1/20 0.32
GSK3B P49841 1/20 0.32
KCNA5 P22460 1/20 0.32
METAP2 P50579 1/20 0.31
CTSA P10619 2/20 0.31
CDC7 O00311 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434756 0.86 CYP3A4 (0.39) GPBAR1CDC7
SCHEMBL9434701 0.85 EGFR (0.40) MAPTCDC7
SCHEMBL9434449 0.85 RPS6KA3 (0.46) GPBAR1MMP13FFAR1ROCK2CDC7
SCHEMBL9433530 0.84 RPS6KA3 (0.35) GPBAR1MMP13CCNCCDK8MAPT
SCHEMBL9434562 0.82 SLC22A12 (0.47) PLCG1CCNCCDK8KCNA5CDC7
SCHEMBL9434742 0.82 GPBAR1 (0.41) PDE4AGPBAR1ROCK2KCNA5
SCHEMBL9433930 0.81 GPBAR1 (0.36) GPBAR1MMP13CCNCCDK8GSK3B
SCHEMBL9433405 0.81 PDE4A (0.43) PDE4AMAPTCDC7
SCHEMBL9433586 0.78 MAOA (0.35) GPBAR1KCNA5
SCHEMBL9433809 0.78 GPBAR1 (0.36) GPBAR1MMP13CCNCCDK8ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed