SCHEMBL9433832

SCHEMBL9433832

COC(=O)C1=C(C)NC(C)=C(c2ccccn2)C1c1ccccc1C#N

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.58
HSD17B10 Q99714 5/20 0.58
CASP1 P29466 3/20 0.48
CASP7 P55210 1/20 0.48
ALDH1A1 P00352 5/20 0.48
HPGD P15428 4/20 0.48
GAA P10253 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
MAPT P10636 2/20 0.44
ADORA3 P0DMS8 2/20 0.44
CACNA1F O60840 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
CACNA1D Q01668 2/20 0.44
KMT2A Q03164 2/20 0.44
CACNA1S Q13698 2/20 0.44
CACNA1C Q13936 2/20 0.44
HIF1A Q16665 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434813 0.88 KDM4E (0.41) KDM4EHSD17B10CASP1CASP7ALDH1A1
SCHEMBL9434085 0.86 KDM4E (0.61) KDM4EHSD17B10CASP1CASP7ALDH1A1
SCHEMBL10432455 0.86 KDM4E (0.64) KDM4EHSD17B10CASP1CASP7ALDH1A1
SCHEMBL7164235 0.84 CYP2C9 (0.59) KDM4EHSD17B10ALDH1A1HPGDGAA
SCHEMBL9433590 0.84 KDM4E (0.61) KDM4EHSD17B10CASP1CASP7ALDH1A1
SCHEMBL9434428 0.84 KDM4E (0.61) KDM4EHSD17B10CASP1CASP7ALDH1A1
SCHEMBL9434613 0.84 KDM4E (0.61) KDM4EHSD17B10CASP1CASP7ALDH1A1
SCHEMBL9434114 0.82 KDM4E (0.81) KDM4EHSD17B10CASP1CASP7ALDH1A1
SCHEMBL9434276 0.82 KDM4E (0.59) KDM4EHSD17B10CASP1CASP7ALDH1A1
SCHEMBL9433816 0.82 CACNA1C (0.46) KDM4EHSD17B10CASP1CASP7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed