SCHEMBL9433877

SCHEMBL9433877

COc1cccc2sc(C(N)=O)c(N)c12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 5/20 0.58
LIMK1 P53667 4/20 0.51
STING1 Q86WV6 2/20 0.48
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 3/20 0.46
GAA P10253 3/20 0.46
HPGD P15428 3/20 0.46
HSD17B10 Q99714 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
GLA P06280 2/20 0.46
MAPK1 P28482 2/20 0.46
TSHR P16473 1/20 0.46
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
MAPT P10636 1/20 0.43
ALOX15 P16050 1/20 0.43
ATM Q13315 1/20 0.43
SLC9A1 P19634 1/20 0.43
BACE1 P56817 1/20 0.42
MAPK3 P27361 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7218005 0.87 KDM4E (0.60) IKBKBSTING1ALDH1A1KDM4EGAA
SCHEMBL9434017 0.81 STING1 (0.46) IKBKBLIMK1STING1ALDH1A1GAA
SCHEMBL3828423 0.80 IKBKB (0.56) IKBKBLIMK1ALDH1A1KDM4EGAA
SCHEMBL20509578 0.76 LIMK1 (0.56) IKBKBLIMK1STING1ALDH1A1KDM4E
SCHEMBL5106264 0.76 IKBKB (0.58) IKBKBLIMK1ALDH1A1KDM4EGAA
SCHEMBL19769187 0.75 IKBKB (0.48) IKBKBLIMK1ALDH1A1KDM4EGAA
SCHEMBL5118198 0.75 IKBKB (0.57) IKBKBLIMK1ALDH1A1KDM4EGAA
SCHEMBL26049804 0.74 EDNRA (0.50) STING1ALDH1A1KDM4EGAAHPGD
SCHEMBL4658241 0.74 IKBKB (1.00) IKBKBLIMK1ALDH1A1KDM4EHPGD
SCHEMBL11101251 0.73 BACE1 (0.54) ALDH1A1KDM4EGAAHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5350748-A 3-thio or amino substituted-benzo[b]thiophene-2-carboxamides and 3-oxygen, thio, or amino substituted-benzofuran-2-carboxamides as inhibitors of cell adhesion WARNER-LAMBERT COMPANY (US) 1994-09-27 US disclosed